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(-)-(alpha)-Kainic Acid (hydrate)
(-)-(alpha)-Kainic Acid (hydrate)

Item number: Cay78050-25

(-)-(alpha)-Kainic acid is a cyclic analog of L-glutamate originally isolated from D. simplex that has neuroexcitatory activities. It binds to the homomeric kainate receptors GluK1, GluK2, GluK3, GluK4, and GluK5 (Kis = 75.9, 12.7, 32.8, 4.7, and 15 nM, respectively). (-)-(alpha)-Kainic acid (5 mM) induces calcium...
Keywords: 2S-carboxy-4S-(1-methylethenyl)-3S-pyrrolidineacetic acid, monohydrate
Application: Central nervous system stimulant
CAS 58002-62-3
MW: 231.2 D
From 97.00€ *
Review
K-Ras(G12C) Inhibitor 9
K-Ras(G12C) Inhibitor 9

Item number: Cay18005-25

K-Ras(G12C) inhibitor 9 is an irreversible, allosteric inhibitor of the K-Ras(G12C) mutant that causes 100% modification of the protein when used at 10 µM for 24 hours in vitro. K-Ras is a small GTPase that cycles between a GTP-bound active state and a GDP-bound inactive state to turn on downstream Raf kinases to...
Keywords: N-[1-[2-[(4-chloro-5-iodo-2-methoxyphenyl)amino]acetyl]-4-piperidinyl]-ethenesulfonamide
Application: KRAS(G12C) inhibitor
CAS 1469337-91-4
MW: 513.8 D
From 60.00€ *
Review