- Search results for Cay70610
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13 products were found matching "Cay70610"!
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Item number: Cay70610-50
Baicalein is a flavonoid originally isolated from the roots of S. baicalensis that has diverse biological activities. It inhibits human platelet 12-lipoxygenase (12-LO) and human reticulocyte 15-LO-1 (IC50s = 0.64 and 1.6 µM, respectively) but is less potent at 15-LO-1 when the detergent Triton-X is present (IC50 =...
Keywords: | 5,6,7-trihydroxyflavone |
Application: | Lipid peroxidation inhibitor |
CAS | 491-67-8 |
MW: | 270.2 D |
From 24.00€
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Item number: Cay70665-10
Arachidonoyl serotonin is an inhibitor of fatty acid amide hydrolase (FAAH), the enzyme responsible for inactivation of anandamide and other endogenous cannabinoids. It inhibits the FAAH activity isolated from mouse neuroblastoma cells with an IC50 value of 12 µM. Both the Km and the Vmax of the enzyme are affected,...
Keywords: | AA-5HT, N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-5Z,8Z,11Z,14Z-eicosatetraenamide |
Application: | FAAH inhibitor |
CAS | 187947-37-1 |
MW: | 462.7 D |
From 66.00€
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Item number: Cay70604-10
3,4-Dihydroxyphenyl ethanol is a phenolic component of olive oil that inhibits both 12- and 5-LO. The IC50 values for the inhibition of rat platelet 12-LO and rat neutrophil 5-LO are 4.2 and 13 µM, respectively. It does not inhibit, and may actually enhance, COX activity. 3,4-Dihydroxyphenyl ethanol also protects...
Keywords: | 3-Hydroxytyrosol, Ba2774, DOPET, 4-(2-hydroxyethyl)-1,2-benzenediol |
Application: | Bioactive lipid assays |
CAS | 10597-60-1 |
MW: | 154.2 D |
From 43.00€
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Item number: Cay70600-10
REV 5901 is an antagonist of cysteinyl-leukotriene receptors with a Ki value of 0.7 µM for guinea pig lung membranes. It is also an inhibitor of rat neutrophil 5-LO with an IC50 value of 0.12 µM.Formal Name: alpha-pentyl-3-(2-quinolinylmethoxy)-benzenemethanol. CAS Number: 101910-24-1. Molecular Formula: C22H25NO2....
Keywords: | alpha-pentyl-3-(2-quinolinylmethoxy)-benzenemethanol |
Application: | 5-LO inhibitor |
CAS | 101910-24-1 |
MW: | 335.4 D |
From 43.00€
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Item number: Cay70660-10
Methyl arachidonyl fluorophosphonate (MAFP) is an inhibitor of monoacylglycerol lipase (MAGL) and fatty acid amide hydrolase (FAAH, IC50s = 26 and 0.33 nM, respectively). It is also an irreversible inhibitor of cytosolic phospholipase A2 (cPLA2), as well as calcium-independent PLA2 (iPLA2, IC50 = 500 nM). MAFP...
Keywords: | MAFP, 5Z,8Z,11Z,14Z-eicosatetraenyl-phosphonofluoridic acid, methyl ester |
Application: | PLA2 inhibitor |
CAS | 188404-10-6 |
MW: | 370.5 D |
From 46.00€
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Item number: Cay70655-10
SC-58125 is a member of the diaryl heterocycle group of selective COX-2 inhibitors which includes MK 966 (rofecoxib), DUP-697, and celecoxib. SC-58125 is a potent and time-dependent inhibitor of COX-2. When tested on the isolated recombinant enzymes, SC-58125 is at least 150 times more potent in the inhibition of...
Keywords: | 5-(4-fluorophenyl)-1-[4-(methylsulfonyl)phenyl]-3-(trifluoromethyl)-1H-pyrazole |
Application: | COX2 inhibitor |
CAS | 162054-19-5 |
MW: | 384.3 D |
From 23.00€
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Item number: Cay70602-10
Caffeic acid is an inhibitor of 5-LO with an IC50 value of 3.7-72 µM and 12-LO with an IC50 value of 5.1-30 µM.Formal Name: 3-(3,4-dihydroxyphenyl)-2-propenoic acid. CAS Number: 331-39-5. Synonyms: 3,4-Dihydroxycinnamic Acid. Molecular Formula: C9H8O4. Formula Weight: 180.2. Purity: >97%. Formulation: (Request...
Keywords: | 3,4-Dihydroxycinnamic Acid, 3-(3,4-dihydroxyphenyl)-2-propenoic acid |
Application: | 5-LO inhibitor |
CAS | 331-39-5 |
MW: | 180.2 D |
From 43.00€
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Item number: Cay70645-10
DuP-697 is a member of the diaryl heterocycle group of selective COX-2 inhibitors which includes MK-966 (rofecoxib), SC-58125, and celecoxib. DuP-697 is a potent and time-dependent inhibitor of COX-2. When tested on isolated recombinant enzymes, DuP-697 is at least 50 times more potent in the inhibition of COX-2...
Keywords: | 5-bromo-2-(4-fluorophenyl)-3-(4-(methylsulfonyl)phenyl)-thiophene |
Application: | COX-2 inhibitor |
CAS | 88149-94-4 |
MW: | 411.3 D |
From 147.00€
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Item number: Cay70690-10
Ketorolac is a non-steroidal anti-inflammatory drug (NSAID) and a non-selective COX inhibitor (IC50 = 20 nM for both COX-1 and COX-2). It prevents increases in paw swelling, increases paw withdrawal latency in a hot-plate test, and decreases prostaglandin E2 (PGE2) levels in paw tissue in a mouse model of...
Keywords: | Toradol, (±)-5-benzoyl-2,3-dihydro-1H-pyrrolizine-1-carboxylic acid, tris(hydroxymethyl)aminomethane salt |
Application: | COX inhibitor |
CAS | 74103-07-4 |
MW: | 376.4 D |
From 61.00€
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Item number: Cay70635-10
Dual cyclooxygenase-2 (COX-2)/5-lipoxygenase (5-LO) inhibitors are potential therapeutic agents for inflammatory diseases and for prostate cancer. CAY10416 is a dual COX-2/5-LO inhibitor with IC50 values of 50 and 3 nM, respectively. The selectivity of CAY10416 for COX is greater than 200-fold for COX-2 versus...
Keywords: | 3-[[3-fluoro-5-(tetrahydro-4-methoxy-2H-pyran-4-yl)phenoxy]methyl]-1-[4-(methylsulfonyl)phenyl]-5-phenyl-1H-pyrazole |
Application: | COX-2 inhibitor, 5-LO inhibitor |
CAS | 443919-96-8 |
MW: | 536.6 D |
From 77.00€
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Item number: Cay70620-10
6-MNA is a competitive, non-selective COX inhibitor. The Ki values for ovine COX-1 and -2 are 21 and 19 µM, respectively. The IC50 values are 70 and 20 µM for human recombinant COX-1 and -2, respectively.Formal Name: 6-methoxy-2-naphthaleneacetic acid. CAS Number: 23981-47-7. Synonyms: 6-MNA. Molecular Formula:...
Keywords: | 6-MNA, 6-methoxy-2-naphthaleneacetic acid |
Application: | COX inhibitor |
CAS | 23981-47-7 |
MW: | 216.2 D |
From 43.00€
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Item number: Cay70664-10
MgammaLnFP is an analog of methyl arachidonyl fluozophosphonate (MAFP, Cay-70660), which has been widely studied as an inhibitor of phospholipases, FAAH, and as a CB receptor ligand. The pharmacology of the gamma-linolenyl analog of MAFP has not been completely investigated.Formal Name:...
Keywords: | MgammaLnFP, 6Z,9Z,12Z-octadecatrienyl-phosphonofluoridic acid, methyl ester |
Application: | FAAH inhibitor |
CAS | 1370451-91-4 |
MW: | 344.4 D |
From 115.00€
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