6 products were found matching "Cay705502-%25"!

Bestatin is an aminopeptidase inhibitor originally isolated from S. olivoreticuli. It inhibits aminopeptidase B (IC50 = 0.05 µg/ml), aminopeptidase N (IC50 = 16.9 µM), leucine aminopeptidase (IC50 = 0.01 µg/ml), and the aminopeptidase activity of leukotriene A4 (LTA4) hydrolase (Kapp = 172 nM). It is selective for...

Ebselen acts as a glutathione peroxidase mimic and is an excellent scavenger of peroxynitrite with a rate constant of 2 x 106 M-1s-1. The glutathione peroxidase-like activity of ebselen inhibits cyclooxygenase and lipoxygenases at micromolar concentrations.Formal Name: 2-phenyl-1,2-benzisoselenazol-3(2H)-one. CAS...

NS 398 is a selective inhibitor of cyclooxygenase-2 (COX-2). The IC50 values for human recombinant COX-1 and -2 are 75 and 1.77 µM, respectively. The IC50 values for ovine COX-1 and -2 are 220 and 0.15 µM, respectively.Formal Name: N-[2-(cyclohexyloxy)-4-nitrophenyl]-methanesulfonamide. CAS Number: 123653-11-2....

1-Benzylimidazole is a selective inhibitor of thromboxane synthase. It reduces TXB2 levels and increases blood flow in ischemia-reperfusion injury of rat brain.Formal Name: 1-(phenylmethyl)-1H-imidazole. CAS Number: 4238-71-5. Molecular Formula: C10H10N2. Formula Weight: 158.2. Purity: >95%. Formulation: (Request...

S-BINOL is a chiral auxiliary for asymmetric ketone reduction, in particular 15-keto prostaglandin intermediates to 15(S)-alcohols.Formal Name: (S)-[1,1'-binaphthalene]-2,2'-diol. CAS Number: 18531-99-2. Synonyms: (S)-BINOL. Molecular Formula: C20H14O2. Formula Weight: 286.3. Purity: >98%. Formulation: (Request...

Fasentin is an inhibitor of glucose transport. It partially inhibits glucose uptake in U937 and DU145 cells when used at concentrations ranging from 15 to 80 µM. Fasentin sensitizes PPC-1 prostate cancer and U937 leukemia cells, but not DU145 prostate cancer cells, to cell death induced by the Fas receptor activator...