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Tolfenamic Acid
Tolfenamic Acid

Item number: Cay70480-25

Tolfenamic acid is a non-steroidal anti-inflammatory drug (NSAID) with anticancer activity. It is selective for COX-2 over COX-1 in canine DH82 monocyte/macrophage cells (IC50s = 3.53 and >51.2 µg/ml, respectively). Tolfenamic acid inhibits calcium influx in human polymorphonuclear leukocytes (PMNLs) induced by...
Keywords: 2-[(3-chloro-2-methylphenyl)amino]-benzoic acid
Application: Nonsteroidal anti-inflammatory drug
CAS 13710-19-5
MW: 261.7 D
From 57.00€ *
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Cambinol
Cambinol

Item number: LKT-C0048.25

Cambinol is an inhibitor of sirtuins, particularly sirtuin1. Cambinol exhibits anti-inflammatory and anticancer chemotherapeutic activities. In various cell lines, cambinol suppresses MAPK and MEK signaling and inhibits expression of pro-inflammatory cytokines such as IL-1 , IL-6, TNF- , and IFN- . Additionally,...
Keywords: SIRT 1/2 inhibitor IV, SIRT1 Inhibitor II, NSC112546, SIRT2 Inhibitor VI.
Application: SIRT1 Inhibitor
CAS 14513-15-6
MW: 360.43 D
From 325.00€ *
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