6 products were found matching "Cay60875-%25"!

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Lumefantrine
Lumefantrine

Item number: Cay20678-25

Lumefantrine is an antimalarial drug that is used in combination with artemether (Cay-11815). The pairing of lumefantrine and artemether is a major form of oral artemisinin combination therapy used against uncomplicated P. falciparum malaria. Lumefantrine also blocks the rapidly activating delayed-rectifier...
Keywords: Benflumetol, CPG-56695, (9Z)-2,7-dichloro-9-[(4-chlorophenyl)methylene]-alpha-[(dibutylamino)methyl]-9H-fluorene-4-methanol
Application: Antimalarial
CAS 82186-77-4
MW: 528.9 D
From 43.00€ *
Review
Clomiphene (citrate)
Clomiphene (citrate)

Item number: Cay16087-25

Clomiphene is a selective estrogen receptor modulator that impairs the activation of estrogen receptors (ERs) by 17beta-estradiol. It potently binds both ERalpha and ERbeta (Ki = 0.9 and 1.2 nM, respectively). Clomiphene enhances the release of gonadotropin-releasing hormone, stimulating the release of...
Keywords: Clomifene, NSC 35770, Omifin, 2-[4-(2-chloro-1,2-diphenylethenyl)phenoxy]-N,N-diethyl-ethanamine...
Application: Selective estrogen receptor modulator
CAS 50-41-9
MW: 598.1 D
From 43.00€ *
Review
Chlorpropamide
Chlorpropamide

Item number: Cay26087-25

Chlorpropamide is a first generation sulfonylurea. It increases glycolysis by increasing fructose-2,6-bisphosphate levels and inhibits glucagon-induced gluconeogenesis by augmenting the effect of insulin in isolated rat hepatocytes when used at a concentration of 0.2 mM. Chlorpropamide reverses increases in blood...
Keywords: NSC 44634, NSC 626720, 4-chloro-N-[(propylamino)carbonyl]-benzenesulfonamide
Application: Antidiabetic, hypoglycemic, sulfonylurea receptor agonist
CAS 94-20-2
MW: 276.7 D
From 92.00€ *
Review
SC-66
SC-66

Item number: Cay10876-25

Akt activation requires binding of its pleckstrin homology domain (PHD) to membrane-associated phosphatidylinositol-3,4,5-trisphosphate (PIP3) or phosphatidylinositol-3,4-bisphosphate (PIP2). Increased Akt activity, e.g., through a gain-of-function mutation in the PHD of Akt1, is pivotal to many types of cancer....
Keywords: 2E,6E-bis(4-pyridinylmethylene)-cyclohexanone
Application: AKT inhibitor
CAS 871361-88-5
MW: 276.3 D
From 52.00€ *
Review
UNC669
UNC669

Item number: Cay10875-25

UNC669 is an inhibitor of the MBT domain of L3MBTL1 with an IC50 value of 6 µM. It is 5- and 10-fold selective for L3MBTL1 over the related proteins L3MBTL3 and L3MBTL4.Formal Name: (5-bromo-3-pyridinyl)[4-(1-pyrrolidinyl)-1-piperidinyl]-methanone. CAS Number: 1314241-44-5. Molecular Formula: C15H20BrN3O. Formula...
Keywords: (5-bromo-3-pyridinyl)[4-(1-pyrrolidinyl)-1-piperidinyl]-methanone
Application: L3MBTL1 antagonist
CAS 1314241-44-5
MW: 338.2 D
From 50.00€ *
Review
Fenpropimorph
Fenpropimorph

Item number: Cay20875-25

Fenpropimorph is a fungicide that inhibits the sterol pathway. It inhibits Delta8-Delta7-sterol isomerase in yeast at low concentrations, with Delta14-sterol reductase being blocked at higher levels, preventing the biosynthesis of ergosterol (Cay-19850). Fenpropimorph is also able to inhibit sterol synthesis in...
Keywords: BAS 42100F, (2R,6S)-rel-4-[3-[4-(1,1-dimethylethyl)phenyl]-2-methylpropyl]-2,6-dimethyl-morpholine
Application: Fungicide, sterol pathway inhibitor
CAS 67564-91-4
MW: 303.5 D
From 109.00€ *
Review