4 products were found matching "Cay360745-%25"!
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TT-232 (trifluoroacetate salt)
Item number: Cay36045-25
TT-232 is a synthetic peptide derivative of somatostatin. It binds to somatostatin receptors in isolated rat synaptosomal membranes (IC50 = ~0.1 nM). TT-232 (30 and 60 µg/ml) inhibits the proliferation of P388 murine and HL-60 human leukemia cells. In vivo, TT-232 (3-12 µg/animal per day) reduces tumor volume in an...
| Keywords: | D-phenylalanyl-L-cysteinyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-cysteinyl-L-threoninamide cyclic (2->6)-disulfide,... |
| Application: | Somatostatin synthetic peptide derivative |
| MW: | 947.1 D |
From 193.00€
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GSK1940029
Item number: Cay36704-25
GSK1940029 is a stearoyl-CoA desaturase (SCD) inhibitor. It increases palmitate-induced phosphorylation of p70 ribosomal S6 kinase 1 (p70S6K1) and lactate dehydrogenase (LDH) release from AML12 hepatocytes when used at a concentration of 20 µM. GSK1940029 (10 µM) also increases palmitate-induced increases in...
| Keywords: | 1-[(3,4-dichlorophenyl)methyl]-N-[4-(hydroxymethyl)phenyl]-5-methyl-1H-1,2,3-triazole-4-carboxamide |
| Application: | Stearoyl-CoA desaturase inhibitor |
| CAS | 1150701-66-8 |
| MW: | 391.3 D |
From 35.00€
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NDI-091143
Item number: Cay36054-25
NDI-091143 is an allosteric inhibitor of ATP citrate lyase (ACL, Ki = 7 nM). It inhibits the production of ADP in a cell-free assay and oxaloacetate production in an enzyme-coupled assay (IC50s = 2.1 and 4.8 nM, respectively).Formal Name:...
| Keywords: | 3-chloro-5-[[(4,6-difluoro[1,1'-biphenyl]-3-yl)amino]sulfonyl]-4-hydroxy-benzoic acid, methyl ester |
| Application: | ACLY inhibitor |
| CAS | 2375840-87-0 |
| MW: | 453.8 D |
From 100.00€
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GSK189254
Item number: Cay36705-25
GSK189254 is a histamine H3 receptor antagonist (Kis = 0.13, 0.68, and 1.74 nM for the recombinant human, rat, and mouse receptors, respectively). It is selective for the histamine H3 receptor over a panel of 50 receptors and ion channels at 1 µM. GSK189254 prevents imetit-induced decreases in forskolin-stimulated...
| Keywords: | GSK189254A, 6-[(3-cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy]-N-methyl-3-pyridinecarboxamide |
| Application: | Histamine H3 receptor antagonist |
| CAS | 720690-73-3 |
| MW: | 351.4 D |
From 147.00€
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