3 products were found matching "Cay18800-%25"!
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6alpha-Methylprednisolone 21-hemisuccinate
Item number: Cay11800-25
6alpha-Methylprednisolone 21-hemisuccinate is a prodrug form of the synthetic glucocorticoid methylprednisolone (Cay-15013). It is converted to methylprednisolone by carboxylesterase 2 (CES2). Nanoliposomes containing 6alpha-methylprednisolone 21-hemisuccinate decreases disease severity in a rat model of...
| Keywords: | 21-(3-carboxy-1-oxopropoxy)-11beta,17-dihydroxy-6alpha-methyl-pregna-1,4-diene-3,20-dione |
| Application: | Inflammation studies |
| CAS | 2921-57-5 |
| MW: | 474.6 D |
From 34.00€
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Felbamate
Item number: Cay18000-25
Felbamate is an inhibitor of NMDA receptors and a modulator of GABAA receptors that also has broad-spectrum inhibitory activity against excitatory amino acid receptors. It binds to NMDA channels with dissociation constants of approximately 200, 110, and 55 µM in the resting, activated, and desensitized states,...
| Keywords: | ADD 03055, 2-phenyl-1,3-propanediol 1,3-dicarbamate |
| Application: | Allosteric NMDA glutamate receptor NR2B subunit antagonist |
| CAS | 25451-15-4 |
| MW: | 238.2 D |
From 60.00€
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ML-264
Item number: Cay18880-25
ML-264 is a selective inhibitor of Krüppel-like factor 5 (KLF5), a zinc finger-containing transcription factor that is highly expressed in rapidly dividing intestinal epithelial cells. It displays an IC50 value of 29 nM in a cell-based assay for proliferation of KLF5-expressing DLD-1 cells and an IC50 value of 81 nM...
| Keywords: | (2E)-3-(3-chlorophenyl)-N-[2-[methyl(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)amino]-2-oxoethyl]-2-propenamide |
| Application: | KLF5 inhibitor |
| CAS | 1550008-55-3 |
| MW: | 384.9 D |
From 43.00€
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