6 products were found matching "Cay171142-%25"!

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OF-1
OF-1

Item number: Cay17124-25

OF-1 is a chemical probe for the bromodomains of the Bromodomain and PHD Finger-containing (BRPF) family of proteins. It binds BRPF1B, BRPF2, and BRPF3 with Kd values of 0.1, 0.5, and 2.4 µM, respectively, as determined by isothermal titration calorimetry. OF-1 increases thermal stability of full length BRPF1B at 1...
Keywords: 4-bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methyl-benzenesulfonamide
Application: BRPF probe
CAS 919973-83-4
MW: 440.3 D
From 66.00€ *
Review
4-P-PDOT
4-P-PDOT

Item number: Cay17411-25

4-P-PDOT is an antagonist of the melatonin 2 (MT2) receptor (pKi = 8.37) that displays 60-fold selectivity for MT2 over MT1. 4-P-PDOT is used in cells, explants, and animals to elucidate the role of MT2 in melatonin-mediated signaling.Formal Name: N-(1,2,3,4-tetrahydro-4-phenyl-2-naphthalenyl)-propanamide. CAS...
Keywords: cis-4-phenyl-2-Propionamidotetralin, AH 024, N-(1,2,3,4-tetrahydro-4-phenyl-2-naphthalenyl)-propanamide
CAS 134865-74-0
MW: 279.4 D
From 89.00€ *
Review
Niclosamide (ethanolamine salt)
Niclosamide (ethanolamine salt)

Item number: Cay17118-25

Niclosamide is a molluscicide. It is toxic to H. trivolvis snail eggs, juveniles, and adults (LC50s = 0.035, 0.044, and 0.11 mg/kg, respectively), as well as rainbow trout, white sucker, and fathead minnow (LC50s = 0.03, 0.09, and 0.11 mg/L, respectively). Niclosamide induces cell cycle arrest at the G0/G1 phase and...
Keywords: BAY-6076, BAY-73, Bayluscide, HL 2448, 5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxy-benzamide compd. with 2-aminoethanol
Application: Anthelmintic, molluscicide
CAS 1420-04-8
MW: 388.2 D
From 36.00€ *
Review
1,25-dihydroxy Vitamin D2
1,25-dihydroxy Vitamin D2

Item number: Cay11174-5

1,25-dihydroxy Vitamin D2 is the active circulating metabolite of vitamin D2 formed by 25-hydroxylase in the liver and 25-hydroxyvitamin D-hydroxylase in the kidney. By binding to the vitamin D receptor (VDR), 1,25-dihydroxy Vitamin D2 activates VDR to interact with the retinoid X receptor (RXR), forming the...
Keywords: Ercalcitriol, Ro 17-6218,...
Application: Metabolic studies
CAS 60133-18-8
MW: 428.7 D
From 121.00€ *
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2-deoxy-2-fluoro L-Fucose
2-deoxy-2-fluoro L-Fucose

Item number: Cay17171-25

2-deoxy-2-fluoro L-Fucose is a fluorinated fucose analog. It can be metabolized inside the cell to a substrate-based inhibitor of fucosyltransferases. Alternatively, it can be converted in vitro to GDP-2-deoxy-2-fluoro L-fucose, a competitive inhibitor of alpha1,3-fucosyltransferase V (Ki = 4.2 µM).Formal Name:...
Keywords: 2,6-dideoxy-2-fluoro-L-galactose
Application: Fucosyltransferase inhibitor
CAS 70763-62-1
MW: 166.1 D
From 60.00€ *
Review
AP219
AP219

Item number: Cay17101-25

AP39 (Cay-17100) is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. It consists of a mitochondria-targeting motif (triphenylphosphonium) coupled to an H2S-donating moiety (dithiolethione) by an aliphatic linker. AP219 is a control compound for AP39, containing the...
Keywords: (9-carboxynonyl)triphenyl-phosphonium
Application: AP39 control
CAS 779282-36-9
MW: 433.6 D
From 43.00€ *
Review