7 products were found matching "Cay16785-%25"!
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15-keto Fluprostenol isopropyl ester
Item number: Cay16786-25
15-keto Fluprostenol isopropyl ester is an ester derivative of the FP receptor agonist fluprostenol (Cay-16768) that is oxidized at carbon 15. It is a potential inactive metabolite of fluprostenol isopropyl ester (travoprost, Cay-16769) based on the published metabolism of latanoprost (Cay-16812) by...
| Keywords: | 15-keto Travoprost,... |
| Application: | Bioactive lipid assays |
| CAS | 404830-45-1 |
| MW: | 498.5 D |
From 118.00€
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2,3-dinor Fluprostenol
Item number: Cay16780-25
2,3-dinor Fluprostenol is a derivative of the FP receptor agonist and prostaglandin F2alpha (PGF2alpha, Cay-16010, Cay-16020) analog fluprostenol (Cay-16768).Formal Name: (+)-9alpha,11alpha,15R-trihydroxy-16-(3-(trifluoromethyl)phenoxy)-2,3,17,18,19,20-hexanor-prosta-5Z,13E-dien-1-oic acid. Molecular Formula:...
| Keywords: | (+)-9alpha,11alpha,15R-trihydroxy-16-(3-(trifluoromethyl)phenoxy)-2,3,17,18,19,20-hexanor-prosta-5Z,13E-dien-1-oic acid |
| Application: | Bioactive lipid assays |
| MW: | 430.4 D |
From 158.00€
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Oxolinic Acid
Item number: Cay16789-25
Bacterial DNA gyrase is a heterodimeric type II topoisomerase that negatively supercoils circular double-stranded DNA. Oxolinic acid is a quinolone antibiotic that inhibits bacterial DNA gyrase, but not eukaryotic topoisomerases, reversibly binding gyrase subunit A in gyrase-DNA complexes, blocking supercoiling...
| Keywords: | NSC 110364, Urinox, 5-ethyl-5,8-dihydro-8-oxo-1,3-dioxolo[4,5-g]quinoline-7-carboxylic acid |
| Application: | Antibiotic, Gyrase inhibitor |
| CAS | 14698-29-4 |
| MW: | 261.2 D |
From 43.00€
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Cryptotanshinone
Item number: Cay16987-25
Cryptotanshinone is a natural quinoid diterpene first isolated from Salvia miltiorrhiza roots, which are used in traditional Chinese medicine for a variety of conditions. Cryptotanshinone, at 10-20 µM, stimulates AMP-activated protein kinase in C2C12 myotubes and activates p38 MAPK in DU145 cells. It inhibits the...
| Keywords: | (1R)-1,2,6,7,8,9-hexahydro-1,6,6-trimethyl-phenanthro[1,2-b]furan-10,11-dione |
| Application: | Apoptosis inducer |
| CAS | 35825-57-1 |
| MW: | 296.4 D |
From 43.00€
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TDZD-8
Item number: Cay16287-25
TDZD-8 is a thiadiazolidine derivative that acts as a non-ATP competitive inhibitor of the serine/threonine kinase glycogen synthase kinase 3beta (GSK3beta, IC50 = 2 µM), binding to the active site of GSK3beta. It does not significantly affect the activities of Cdk-1/cyclin B, CK-II, cAMP-dependent protein kinase,...
| Keywords: | GSK3beta Inhibitor I, NP 01139, 2-methyl-4-(phenylmethyl)-1,2,4-thiadiazolidine-3,5-dione |
| Application: | GSK3-beta inhibitor |
| CAS | 327036-89-5 |
| MW: | 222.3 D |
From 82.00€
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Clomiphene (citrate)
Item number: Cay16087-25
Clomiphene is a selective estrogen receptor modulator that impairs the activation of estrogen receptors (ERs) by 17beta-estradiol. It potently binds both ERalpha and ERbeta (Ki = 0.9 and 1.2 nM, respectively). Clomiphene enhances the release of gonadotropin-releasing hormone, stimulating the release of...
| Keywords: | Clomifene, NSC 35770, Omifin, 2-[4-(2-chloro-1,2-diphenylethenyl)phenoxy]-N,N-diethyl-ethanamine... |
| Application: | Selective estrogen receptor modulator |
| CAS | 50-41-9 |
| MW: | 598.1 D |
From 43.00€
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Hemin chloride
Item number: Cay16487-25
Hemin chloride is an oxidized form of heme that inhibits eukaryotic translation initiation factor 2alpha kinase 1 (eIF2alphaK1), a repressor of eIF-2alpha. This alters the initiation of mRNA translation, evoking a wide array of cellular effects. Hemin chloride is used experimentally to induce the expression of heme...
| Keywords: | (SP-5-13)-chloro[7,12-diethenyl-3,8,13,17-tetramethyl-21H,23H-porphine-2,8-dipropanoato(4-)-kappaN21, kappaN22, kappaN23,... |
| Application: | EIF2AK1 inhibitor |
| CAS | 16009-13-5 |
| MW: | 652 D |
From 66.00€
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