5 products were found matching "Cay16120"!
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Prostaglandin F2alpha 1,15-lactone
Item number: Cay16120-5
Prostaglandin F2alpha (PGF2alpha) 1,15-lactone is a lipid-soluble internal ester of PGF2alpha. Hydrolysis of the lactone readily produces free PGF2alpha in plasma. In rhesus monkeys, a total dose of 15 mg of PGF2alpha 1,15-lactone terminates early pregnancy, whereas PGF2alpha is ineffective.Formal Name:...
| Keywords: | PGF2alpha 1,15-lactone, 9alpha,11alpha,15S-trihydroxy-prosta-5Z,13E-dien-1-oic acid, 1,15-lactone |
| Application: | Bioactive lipid assays |
| CAS | 55314-49-3 |
| MW: | 336.5 D |
From 117.00€
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7-Ethoxyresorufin
Item number: Cay16122-10
7-Ethoxyresorufin (7-ER) is a fluorogenic substrate for, and competitive inhibitor of, the cytochrome P450 (CYP) isoform CYP1A1 (IC50 = 0.1 µM). Upon enzymatic cleavage by CYP1A1, resorufin is released and its fluorescence can be used to quantify CYP1A1 activity. Resorufin displays excitation/emission maxima of...
| Keywords: | 7-ER, 7-Ethoxyphenoxazone, Resorufin ethyl ether, 7-ethoxy-3H-phenoxazin-3-one |
| Application: | Cytochrome P450 1A1 fluorometric substrate / competitive inhibitor |
| CAS | 5725-91-7 |
| MW: | 241.2 D |
From 77.00€
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Levosimendan
Item number: Cay16128-50
Levosimendan is a calcium sensitizer that can cause increased cardiac contractility by binding troponin C (EC50 = 9 nM), promotes vasodilation by activating ATP-sensitive potassium channels on vascular smooth muscle cells (EC50 = 0.28 µM), and performs a cardioprotective function by prompting the opening of...
| Keywords: | (R)-Simendan, OR 1259, Simdax(R),... |
| Application: | PDE3 inhibitor |
| CAS | 141505-33-1 |
| MW: | 280.3 D |
From 77.00€
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(±)4-Hydroxymephenytoin
Item number: Cay16124-10
(±)4-Hydroxymephenytoin is a metabolite of (R)-mephenytoin (Cay-25891) and (S)-mephenytoin (Cay-11913). It is formed from (R)- and (S)-mephenytoin by the cytochrome P450 (CYP) isoform CYP2C19 in the liver.Formal Name: 5-ethyl-5-(4-hydroxyphenyl)-3-methyl-2,4-imidazolidinedione. CAS Number: 61837-65-8. Molecular...
| Keywords: | 5-ethyl-5-(4-hydroxyphenyl)-3-methyl-2,4-imidazolidinedione |
| Application: | (S)-mephenytoin metabolite |
| CAS | 61837-65-8 |
| MW: | 234.3 D |
From 142.00€
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DIDS (sodium salt)
Item number: Cay16125-50
DIDS is a stilbene sulfonate that inhibits anionic transport. It has been used to inhibit Cl- uptake through plasma membrane-localized Cl- channels in order to study chloride transport. It also effectively inhibits various sodium-coupled bicarbonate transporters.Formal Name:...
| Keywords: | 4,4'-Diisothiocyanato-2.2'-stilbenedisulfonic acid, MDL 101114ZA,... |
| Application: | Anionic transport inhibitor |
| CAS | 67483-13-0 |
| MW: | 498.5 D |
From 60.00€
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