4 products were found matching "Cay160780-%25"!
No results were found for the filter!
2,3-dinor Fluprostenol
Item number: Cay16780-25
2,3-dinor Fluprostenol is a derivative of the FP receptor agonist and prostaglandin F2alpha (PGF2alpha, Cay-16010, Cay-16020) analog fluprostenol (Cay-16768).Formal Name: (+)-9alpha,11alpha,15R-trihydroxy-16-(3-(trifluoromethyl)phenoxy)-2,3,17,18,19,20-hexanor-prosta-5Z,13E-dien-1-oic acid. Molecular Formula:...
| Keywords: | (+)-9alpha,11alpha,15R-trihydroxy-16-(3-(trifluoromethyl)phenoxy)-2,3,17,18,19,20-hexanor-prosta-5Z,13E-dien-1-oic acid |
| Application: | Bioactive lipid assays |
| MW: | 430.4 D |
From 158.00€
*
Clomiphene (citrate)
Item number: Cay16087-25
Clomiphene is a selective estrogen receptor modulator that impairs the activation of estrogen receptors (ERs) by 17beta-estradiol. It potently binds both ERalpha and ERbeta (Ki = 0.9 and 1.2 nM, respectively). Clomiphene enhances the release of gonadotropin-releasing hormone, stimulating the release of...
| Keywords: | Clomifene, NSC 35770, Omifin, 2-[4-(2-chloro-1,2-diphenylethenyl)phenoxy]-N,N-diethyl-ethanamine... |
| Application: | Selective estrogen receptor modulator |
| CAS | 50-41-9 |
| MW: | 598.1 D |
From 43.00€
*
SR 3677
Item number: Cay16708-25
SR 3677 is a potent, ATP-competitive inhibitor of Rho-associated kinases (ROCKs) that shows greater potency against ROCK2 than ROCK1 in enzyme and cell-based assays (IC50 values are 3 and 56 nM, respectively). At 3 µM, SR 3677 inhibits only 5 (Akt3, Clk1, Clk2, Clk4, Lats2) out of 353 kinases with greater than 50%...
| Keywords: | N-[2-[2-(dimethylamino)ethoxy]-4-(1H-pyrazol-4-yl)phenyl]-2,3-dihydro-1,4-benzodioxin-2-carboxamide |
| Application: | ROCK inhibitor |
| CAS | 1072959-67-1 |
| MW: | 408.5 D |
From 60.00€
*
R-7050
Item number: Cay16870-25
R-7050 is a cell-permeable antagonist of signaling through the TNF-alpha receptor complex (EC50 = 0.631 µM). It blocks TNF-alpha-induced binding of TNF-alpha receptor I with TNF-alpha receptor-associated death domain protein and receptor interacting protein 1, which, in turn, prevents internalization of the receptor...
| Keywords: | TNF-alpha Antagonist III, 8-chloro-4-(phenylthio)-1-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]quinoxaline |
| Application: | Cell-permeable TNF-alpha receptor complex signaling antagonist |
| CAS | 303997-35-5 |
| MW: | 380.8 D |
From 43.00€
*
