- Search results for Cay15010
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14 products were found matching "Cay15010"!
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Item number: Cay15010-1
Prostaglandin F1alpha (PGF1alpha) is the putative metabolite of dihomo-gamma-linolenic acid (DGLA) via the cyclooxygenase (COX) pathway. Both PGF1alpha and PGF2alpha (Cay-16010, Cay-10007221) have been shown to act as priming pheromones for male Atlantic salmon with a threshold concentration of 10-11 M. PGF1alpha...
Keywords: | PGF1alpha, 9alpha,11alpha,15S-trihydroxy-prost-13E-en-1-oic acid |
Application: | Bioactive lipid assays |
CAS | 745-62-0 |
MW: | 356.5 D |
From 74.00€
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Item number: Cay11500-10
ABT-263 is an inhibitor of the Bcl-2 family proteins Bcl-2, Bcl-xL, and Bcl-W (Kis = is = 550 and 354 nM, respectively). ABT-263 is cytotoxic in a panel of small cell lung cancer (SCLC), leukemia, and lymphoma cell lines with a mean EC50 value of 1 µM. It induces apoptosis in influenza A-infected retinal pigment...
Keywords: | A-855071, Navitoclax,... |
Application: | Potent, cell-permeable BH3 domain mimetic |
CAS | 923564-51-6 |
MW: | 974.6 D |
From 33.00€
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Item number: Cay11550-10
5-Methoxy-N,N-diisopropyltryptamine (5-MeO DiPT) (Cay-11865) is a psychedelic hallucinogen which is abused worldwide. Known informally as 'foxy', this compound potently inhibits the re-uptake of dopamine, serotonin, and norepinephrine (IC50s = 65, 2.2, and 8.2 µM, respectively). DiPT is an uncommonly abused...
Keywords: | N,N-Diisopropyltryptamine, N,N-bis(1-methylethyl)-1H-indole-3-ethanamine |
Application: | Analytical reference standard, Uncommonly abused psychedelic drug related to 5-MeO DiPT |
CAS | 14780-24-6 |
MW: | 244.4 D |
From 258.00€
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Item number: Cay15550-10
Mammalian Omi/HtrA2 is a serine protease localized in mitochondria with close homology to bacterial HtrA chaperones. It is released from the mitochondria in response to apoptotic stimuli whereupon it induces cell death through both a caspase-dependent manner and a mechanism that involves its protease activity. UCF...
Keywords: | dihydro-5-[[5-(2-nitrophenyl)-2-furanyl]methylene]-1,3-diphenyl-2-thioxo-4,6(1H,5H)-pyrimidinedione |
Application: | OMI / HTRA2 inhibitor |
CAS | 313649-08-0 |
MW: | 495.5 D |
From 48.00€
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Item number: Cay15055-10
ADB-PINACA (Cay-14763) is an analog of AKB48 (Cay-ISO00060), the pentyl indazole with structural similarity to JWH 018 adamantyl carboxamide (Cay-9001193) and STS-135 (Cay-11564), which are synthetic cannabinoids (CBs) with potential to be sold for recreational abuse. ADB-PINACA pentanoic acid metabolite is an...
Keywords: | 3-[[[1-(aminocarbonyl)-2,2-dimethylpropyl]amino]carbonyl]-1H-indazole-1-pentanoic acid |
Application: | Analytical reference standard, Expected major ADB-PINACA phase I metabolite |
CAS | 2460433-29-6 |
MW: | 374.4 D |
From 158.00€
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Item number: Cay15037-10
Mibefradil is a general calcium channel blocker that shows modest selectivity for T-type channels over L-type channels (IC50 = 2.7 and 18.6 µM, respectively). It is a potent vasodilator, increasing coronary artery flow with an EC50 value of 54 nM. Mibefradil has minimal negative inotropic effects, supporting its use...
Keywords: | Posicor, Ro 40-5967,... |
Application: | Calcium channel blocker, Vasodilator |
CAS | 116666-63-8 |
MW: | 568.6 D |
From 142.00€
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Item number: Cay15045-10
Dofetilide is a class III antiarrhythmic agent that prolongs cardiac action potential duration by selectively inhibiting the rapidly activating inward rectifying component of net delayed rectifier K+ current (IC50 = 31.5 nM in guinea pig cardiomyocytes). However, at 1 µM, dofetilide has pro-arrhythmic activity,...
Keywords: | Tikosyn, UK 68789, N-[4-[2-[methyl[2-[4-[(methylsulfonyl)amino]phenoxy]ethyl]amino]ethyl]phenyl]-methanesulfonamide |
Application: | Voltage-gated potassium channel (KCNH2) blocker |
CAS | 115256-11-6 |
MW: | 441.6 D |
From 84.00€
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Item number: Cay15027-10
Tolterodine is an antagonist of muscarinic acetylcholine receptors (Kis = 1.4, 2.7, 3.6, 3.1, and 2.2 nM for M1-5 receptors, respectively). It reduces intracellular calcium mobilization induced by carbachol (carbamoylcholine, Cay-14486) in bladder smooth muscle cells and submandibular gland cells isolated from...
Keywords: | PNU 200583E, 2-[(1R)-3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-methyl-phenol, 2R,3R-dihydroxybutanedioate |
Application: | Muscarinic (M) receptor antagonist |
CAS | 124937-52-6 |
MW: | 475.6 D |
From 115.00€
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Item number: Cay15035-10
Cilostazol is a phosphodiesterase 3A (PDE3A) inhibitor (IC50 = 0.2 µM for the platelet enzyme). It is selective for PDE3A over PDE1, -2, -4, and -5 (IC50s = >5 µM for all). Cilostazol inhibits collagen- or ADP-induced aggregation of isolated rabbit platelets (IC50s = 29 and 31 µM, respectively). In vivo, cilostazol...
Keywords: | OPC 13013, OPC 21, Pletaal, Pletal, 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone |
Application: | PDE3 inhibitor |
CAS | 73963-72-1 |
MW: | 369.5 D |
From 40.00€
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Item number: Cay15031-10
Ziprasidone is an atypical antipsychotic. It is an agonist of the serotonin (5-HT) receptor subtype 5-HT1A (EC50 = 36.31 nM for inhibition of forskolin-induced adenylate cyclase activity in HeLa cells expressing human receptors), as well as an inverse agonist of 5-HT1D receptors (IC50 = 2.69 nM) and a partial...
Keywords: | CP-88,059, 5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-2H-indol-2-one, monohydrochloride,... |
Application: | Serotonin 5-HT2A and dopamine D2 antagonist, 5-HT1A receptor agonist |
CAS | 138982-67-9 |
MW: | 467.4 D |
From 60.00€
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Item number: Cay15038-10
Reboxetine is an antidepressant compound that selectively inhibits norepinephrine uptake (IC50s = 8.2 and 1,070 nM for norepinephrine and serotonin transporters, respectively). It displays greater than 1,000-fold affinity for binding rat norepinephrine receptors compared to serotonin, histamine, acetylcholine, or...
Keywords: | Davedax, Edronax, FCE 20124, PNU 155950E, (2R)-rel-2-[(R)-(2-ethoxyphenoxy)phenylmethyl]-morpholine, methanesulfonate |
Application: | Norepinephrine uptake inhibitor, Noradrenalin transporter inhibitor |
CAS | 98769-84-7 |
MW: | 409.5 D |
From 84.00€
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Item number: Cay15005-10
Bazedoxifene (acetate) is a third generation selective estrogen receptor modulator (SERM). It is an indole-based ER ligand that binds to both ERalpha (IC50 = 26 nM) and ERbeta (IC50 = 99 nM). Bazedoxifene (actetate) antagonizes 17beta-estradiol-dependent MCF-7 and T47D breast cancer cell proliferation in vitro as...
Keywords: | TSE 424, 1-[[4-[2-(hexahydro-1H-azepin-1-yl)ethoxy]phenyl]methyl]-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-ol, acetate |
Application: | Selective estrogen receptor modulator |
CAS | 198481-33-3 |
MW: | 530.7 D |
From 149.00€
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