19 products were found matching "Cay14910"!

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19(R)-hydroxy Prostaglandin E2
19(R)-hydroxy Prostaglandin E2

Item number: Cay14910-50

19(R)-hydroxy Prostaglandin E2 (19(R)-hydroxy PGE2) is found in the semen of primates, including man. It is a potent smooth muscle relaxant and a selective agonist for the EP2 receptor. It has an EC50 value of 200 nM for relaxing cat tracheal rings which express EP2 receptors.Formal Name:...
Keywords: 19(R)-hydroxy PGE2, 19(R)-OH PGE2, 9-oxo-11alpha,15S,19R-trihydroxy-prosta-5Z,13E-dien-1-oic acid
Application: EP2 receptor agonist
CAS 64625-54-3
MW: 368.5 D
From 76.00€ *
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Blasticidin S (hydrochloride)
Blasticidin S (hydrochloride)

Item number: Cay14499-10

Blasticidin S is a peptidyl nucleoside antibiotic. It was first isolated from S. griseochromogenes. The structure of the pentahydrate form was determined using diffractometer data and, similar to the antibiotic amicetin, the hydrophilic and hydrophobic groups lie on either side of the molecule. It has since been...
Keywords: 4-[[(3S)-3-amino-5-[(aminoiminomethyl)methylamino]-1-oxopentyl]amino]-1-(4-amino-2-oxo-1(2H)-pyrimidinyl)-1,2,3,4-tetradeo...
Application: Antibiotic
CAS 3513-03-9
MW: 458.9 D
From 54.00€ *
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Obatoclax (mesylate)
Obatoclax (mesylate)

Item number: Cay11499-10

Obatoclax is an antagonist of Bcl-2 family members containing four Bcl-2 homology domains, including Bcl-2, Bcl-W, Bcl-xL, and Mcl-1 (Kd = ~500 nM). It prevents the interaction of these pro-survival proteins with Bax or Bak, thereby inducing apoptosis with up-regulation of Bim, induced cytochrome c release, and...
Keywords: GX15-070, 2-[2-[(3,5-dimethyl-1H-pyrrol-2-yl)methylene]-3-methoxy-2H-pyrrol-5-yl]-1H-indole, monomethanesulfonate
Application: Antagonist of Bcl-2 family members containing four Bcl-2 homology domains
CAS 803712-79-0
MW: 413.5 D
From 84.00€ *
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Ondansetron (hydrochloride hydrate)
Ondansetron (hydrochloride hydrate)

Item number: Cay14999-10

Ondansetron (hydrochloride hydrate) (Cay-14999) is an analytical reference material categorized as an antiemetic. Formulations containing ondansetron have been used to reduce alcohol consumption and mood disturbances in early-onset alcoholics. This product is intended for research and forensic applications.Formal...
Keywords: Emeset, GR 38032F, NSC 665799, SN 307,...
Application: Analytical reference material, Serotonin 5-HT3 receptor antagonist, Antiemetic
CAS 103639-04-9
MW: 365.9 D
From 146.00€ *
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Tetrahydroharmine
Tetrahydroharmine

Item number: Cay14449-10

Tetrahydroharmine (THH) is a fluorescent indole alkaloid extracted from B. caapi, a woody vine that is used to produce a psychoactive beverage, ayahuasca, which has been ritually ingested for medicoreligious purposes throughout South America since pre-Columbian times. THH inhibits monoamine oxidase (MAO)-A and MAO-B...
Keywords: Leptaflorine, THH, 2,3,4,9-tetrahydro-7-methoxy-1-methyl-1H-pyrido[3,4-b]indole
Application: MAO inhibitor
CAS 17019-01-1
MW: 216.3 D
From 62.00€ *
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Pyrazolam
Pyrazolam

Item number: Cay14901-10

Pyrazolam is a benzodiazepine that has been abused recreationally. Like other benzodiazepines, pyrazolam has anxiolytic effects. This product is intended for forensic and research purposes.Formal Name: 8-bromo-1-methyl-6-(2-pyridinyl)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine. CAS Number: 39243-02-2. Molecular...
Keywords: 8-bromo-1-methyl-6-(2-pyridinyl)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine
Application: Analytical reference standard, Recreationally abused Benzodiazepine
CAS 39243-02-2
MW: 354.2 D
From 291.00€ *
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Nitracaine
Nitracaine

Item number: Cay14900-10

Nitracaine is a structural analog of dimethocaine, a local anesthetic that inhibits dopamine reuptake through the dopamine transporter and is characterized by reinforcing behavioral effects in rhesus monkey similar to that of cocaine. The physiological and toxicological properties of this compound are not known....
Keywords: 3-(diethylamino)-2,2-dimethylpropyl 4-nitrobenzoate
Application: Analytical reference material, Structural dimethocaine analog
CAS 1648893-21-3
MW: 308.4 D
From 84.00€ *
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Paroxetine (hydrochloride)
Paroxetine (hydrochloride)

Item number: Cay14998-10

Paroxetine is a selective serotonin reuptake inhibitor (SSRI, Ki = 0.04 nM). It is selective for the serotonin transporter (SERT) over the dopamine and norepinephrine transporters (Kis = 400 and 90 nM, respectively) as well as the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT2A, the histamine H1 receptor,...
Keywords: BRL 29060A, (3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-fluorophenyl)-piperidine, monohydrochloride
Application: Serotonin reuptake inhibitor
CAS 78246-49-8
MW: 365.8 D
From 66.00€ *
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NBQX (sodium salt)
NBQX (sodium salt)

Item number: Cay14914-50

Ionotropic glutamate receptors can be divided into three groups, depending on whether they are activated by alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA), kainate, or N-methyl-D-aspartate (NMDA). NBQX is a water-soluble receptor antagonist which targets both AMPA- and kainate-sensitive glutamate...
Keywords: 1,2,3,4-tetrahydro-6-nitro-2,3-dioxo-benzo[f]quinoxaline-7-sulfonamide, disodium salt
Application: AMPA / kainate-sensitive glutamate receptor antagonist
CAS 479347-86-9
MW: 380.2 D
From 149.00€ *
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Arctigenin
Arctigenin

Item number: Cay14913-10

Arctigenin is an extract from A. lappa, a burdock plant traditionally used in Japanese Kampo medicine for its antioxidant, anti-inflammatory, antiproliferative, and antiviral activity. At 0.1 µM, arctigenin can block the activation of Akt induced by glucose starvation in pancreatic cancer PANC-1 cells, which is a...
Keywords: (3R,4R)-4-[(3,4-dimethoxyphenyl)methyl]dihydro-3-[(4-hydroxy-3-methoxyphenyl)methyl]-2(3H)-furanone
Application: Antiviral agent
CAS 7770-78-7
MW: 372.4 D
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24-dehydro Cholesterol
24-dehydro Cholesterol

Item number: Cay14943-10

24-dehydro Cholesterol is an immediate precursor to cholesterol in the Bloch pathway of cholesterol biosynthesis. Structurally, it varies from cholesterol only by a single double bond at carbon 24 and has been used as cholesterol substitute in cellular membrane studies. During brain development, 24-dehydro...
Keywords: Desmosterol, NSC 226126, (3beta)-cholesta-5,24-dien-3-ol
Application: Cholesterol precursor
CAS 313-04-2
MW: 384.6 D
From 48.00€ *
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LMK 235
LMK 235

Item number: Cay14969-10

Histone deacetylases (HDACs) catalyze the hydrolytic removal of acetyl groups from histone lysine residues, which commonly results in chromatin condensation and transcriptional repression. LMK 235 is an HDAC inhibitor that selectively targets HDACs 4 and 5 (IC50s = 12 and 4 nM, respectively) over other HDACs (IC50s...
Keywords: N-[[6-(hydroxyamino)-6-oxohexyl]oxy]-3,5-dimethyl-benzamide
Application: HDAC4 inhibitor, HDAC5 inhibitor
CAS 1418033-25-6
MW: 294.4 D
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