3 products were found matching "Cay13756-%25"!
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Isradipine
Item number: Cay17536-25
Isradipine is a selective L-type calcium channel blocker with long-acting antihypertensive activity. It demonstrates an EC50 value of 1.4 nM for relaxation of depolarization-induced contractions of rabbit aorta and an EC25 value of 0.45 nM for reduction in rate of spontaneously beating guinea pig right atria. By...
| Keywords: | PN 200-110, 4-(2,1,3-benzoxadiazol-4-yl)-1,4-dihydro-2,6-dimethyl-3,5-pyridinedicarboxylic acid, 3-methyl... |
| Application: | L-type calcium channel blocker |
| CAS | 75695-93-1 |
| MW: | 371.4 D |
From 60.00€
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WP1066
Item number: Cay14736-25
WP1066 is a cell-permeable inhibitor of STAT3 that directs dephosphorylation and nuclear export of constitutively phosphorylated STAT3 in U87-MG and U373-MG malignant glioma cells when given at a concentration of 10 µM. It also induces apoptosis in U87-MG (IC50 = 5.6 µM) and U373-MG (IC50 = 3.7 µM) cells. WP1066 is...
| Keywords: | STAT Inhibitor III, 3-(6-bromo-2-pyridinyl)-2-cyano-N-[(1S)-1-phenylethyl]-2E-propenamide |
| Application: | STAT3 inhibitor |
| CAS | 857064-38-1 |
| MW: | 356.2 D |
From 43.00€
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(±)-WIN 55,212 (mesylate)
Item number: Cay10736-25
(±)-WIN 55,212 is a racemic mixture of the cannabinoid (CB) receptor 1 (CB1) and CB2 agonist (+)-WIN 55,212-2 (Cay-10009023) and the CB2 neutral antagonist (-)-WIN 55,212-3 (Cay-12022). It inhibits electrically induced contractions in mouse vas deferens preparations (IC50 = 0.006 µM) and reduces prostaglandin (PG)...
| Keywords: | [2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanone,... |
| Application: | CB receptor agonist |
| CAS | 137795-17-6 |
| MW: | 522.6 D |
From 56.00€
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