4 products were found matching "Cay13706-%25"!
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(±)-WIN 55,212 (mesylate)
Item number: Cay10736-25
(±)-WIN 55,212 is a racemic mixture of the cannabinoid (CB) receptor 1 (CB1) and CB2 agonist (+)-WIN 55,212-2 (Cay-10009023) and the CB2 neutral antagonist (-)-WIN 55,212-3 (Cay-12022). It inhibits electrically induced contractions in mouse vas deferens preparations (IC50 = 0.006 µM) and reduces prostaglandin (PG)...
| Keywords: | [2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanone,... |
| Application: | CB receptor agonist |
| CAS | 137795-17-6 |
| MW: | 522.6 D |
From 56.00€
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SB-224289 (hydrochloride)
Item number: Cay17036-25
The transduction of neurobehavioral effects by serotonin (5-hydroxy tryptamine, 5-HT) is mediated by at least seven major 5-HT receptor subtypes. SB-224289 is a potent 5-HT1B inverse agonist (pKi = 8.16) that displays >75-fold selectivity for human 5-HT1B over all other 5-HT receptors. It has been used to study the...
| Keywords: | [2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl](2,5,6,7-tetrahydro-1'-methylspiro[3H-furo[2,3-f]indole-... |
| Application: | 5-HT1B inverse agonist |
| CAS | 180084-26-8 |
| MW: | 557.1 D |
From 77.00€
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Laurdan
Item number: Cay19706-25
Laurdan is a membrane-permeable fluorescent probe that displays spectral sensitivity to the phospholipid phase of the cell membrane to which it is bound. Quantitation of generalized polarization (GP) of laurdan can be used to identify phospholipid phase. When excited at 340 nm, GP values are 0.6 and -0.2 for gel...
| Keywords: | 1-[6-(dimethylamino)-2-naphthalenyl]-1-dodecanone |
| Application: | Membrane permeable fluorescent probe, GP quantitation |
| CAS | 74515-25-6 |
| MW: | 353.5 D |
From 64.00€
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VU0155069
Item number: Cay13206-25
Phospholipase D (PLD) is an enzyme which cleaves the head group from phospholipids, producing the second messenger phosphatidic acid. Two mammalian isoforms of PLD, PLD1 and PLD2, have been identified, with multiple splice variants of each. Although the two isoforms share structural and functional features, they are...
| Keywords: | CAY10593, N-[2-[4-(5-chloro-2,3-dihydro-2-oxo-1H-benzimidazol-1-yl)-1-piperidinyl]-1-methylethyl]-2-naphthalenecarboxamide |
| Application: | PLD1 inhibitor |
| MW: | 463 D |
From 50.00€
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