4 products were found matching "Cay13612-%25"!
No results were found for the filter!
Pristimerin
Item number: Cay13621-25
Monoacylglycerol lipase (MAGL) hydrolyzes the endogenous cannabinoid 2-arachidonoyl glycerol (2-AG), terminating its capacity to activate cannabinoid receptors. Pristimerin is a naturally occurring terpenoid that potently inhibits MAGL (IC50 = 93 nM). Its actions are rapid, reversible, and noncompetitive....
| Keywords: | Celastrol methyl ester, NSC 99281, 3-hydroxy-9beta,13alpha-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic... |
| Application: | Monoacylglycerol lipase inhibitor |
| CAS | 1258-84-0 |
| MW: | 464.6 D |
From 130.00€
*
ACS 67
Item number: Cay13619-25
Latanoprost is an F-series prostaglandin (PG) analog which has been approved for use as an ocular hypotensive drug for the treatment of glaucoma. Latanoprost is an isopropyl ester, a prodrug form which is converted to latanoprost (free acid) by endogenous esterase enzymes. The free acid form is 200 times more potent...
| Keywords: | 7-[(1R,2R,3R,5S)-3,5-dihydroxy-2-[(3R)-3-hydroxy-5-phenylpentyl]cyclopentyl]-4-(3-thioxo-3H-1,2-dithiol-5-yl)phenyl ester,... |
| Application: | Latanoprost analog |
| CAS | 1088434-86-9 |
| MW: | 598.8 D |
From 105.00€
*
URB447
Item number: Cay13261-25
URB447 is a cannabinoid 1 (CB1) receptor antagonist and CB2 receptor agonist. It inhibits the binding of the CB receptor agonist [3H]-WIN 55,212-2 to CHO-K1 cells expressing the human CB2 receptor or rat cerebellar membranes (IC50s = 41 and 313 nM, respectively). URB447 (20 mg/kg) reduces food intake and weight gain...
| Keywords: | [4-amino-1-[(4-chlorophenyl)methyl]-2-methyl-5-phenyl-1H-pyrrol-3-yl]phenyl-methanone |
| Application: | CB1 receptor antagonist, CB2 receptor agonist |
| CAS | 1132922-57-6 |
| MW: | 400.9 D |
From 110.00€
*
Ibandronate (sodium hydrate)
Item number: Cay21361-25
Ibandronate is a bisphosphonate that has been used in formulations for the treatment of osteoporosis. It binds to hydroxyapatite crystals with an affinity constant of 2.36 µM, inhibiting their growth and bone resorption.Formal Name: P,P'-[1-hydroxy-3-(methylpentylamino)propylidene]bis-phosphonic acid, monosodium...
| Keywords: | P,P'-[1-hydroxy-3-(methylpentylamino)propylidene]bis-phosphonic acid, monosodium salt, monohydrate |
| Application: | Bisphosphonate, osteoporosis agent, FDPS inhibitor |
| CAS | 138926-19-9 |
| MW: | 359.2 D |
From 54.00€
*
