- Search results for Cay13539-%25
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8 products were found matching "Cay13539-%25"!
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COVID-19 Research
Item number: Cay13533-25
E-64d is an irreversible, membrane-permeable inhibitor of lysosomal and cytosolic cysteine proteases and has diverse biological activities. It is a synthetic analog of E-64 (Cay-10007963) and prodrug form of E-64c (Cay-10007964) that inhibits calpain and the cysteine proteases cathepsins F, -K, -B, -H, and...
Keywords: | Aloxistatin, E-64c ethyl ester, EP 453, EST, Loxistatin, NSC 694281,... |
Application: | Protease inhibitor |
CAS | 88321-09-9 |
MW: | 342.4 D |
From 66.00€
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Item number: Cay13531-25
(-)-Warfarin is a component of (±)-warfarin (Cay-13566). It is an anticoagulant that interferes with interconversion of vitamin K and vitamin K epoxide and the role of vitamin K in carboxylation of several clotting cascade proteins, inhibiting the initiation of clotting. In vivo, (-)-warfarin slows formation of the...
Keywords: | (S)-Warfarin, 4-hydroxy-3-[(1S)-3-oxo-1-phenylbutyl]-2H-1-benzopyran-2-one |
Application: | Anti-coagulant |
CAS | 5543-57-7 |
MW: | 308.3 D |
From 94.00€
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Item number: Cay15393-25
BQCA is a highly selective positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR), as it dose-dependently reduces the concentration of acetylcholine required to activate the M1 receptor. The effective range for potentiation of M1 in cells by BQCA is 0.1 to 100 µM with an inflection point...
Keywords: | 1,4-dihydro-1-[(4-methoxyphenyl)methyl]-4-oxo-3-quinolinecarboxylic acid |
Application: | Highly selective positive allosteric muscarinic acetylcholine receptor M1 modulator |
CAS | 338747-41-4 |
MW: | 309.3 D |
From 84.00€
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Item number: Cay13139-25
Imatinib is an inhibitor of the receptor tyrosine kinases c-Abl, Bcr-Abl, PDGFR, and c-Kit. It inhibits ligand-stimulated autophosphorylation of PDGFR and c-Kit (IC50s = ~0.3 and ~0.1 µM, respectively). Imatinib inhibits the proliferation of Bcr-Abl-dependent R10(-) cells (IC50s = ~35-40 nM) and HMC-1 cells...
Keywords: | CGP57148B, STI-571,... |
Application: | Tyrosine kinase inhibitor |
CAS | 220127-57-1 |
MW: | 589.7 D |
From 40.00€
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Item number: Cay10539-50
Very long chain polyunsaturated fatty acids (VLCPUFAs) are important components of ceramides and sphingomyelin and are present in retina, sperm, and brain. Tetratriaconta-16(Z),19(Z),22(Z),25(Z),28(Z),31(Z)-hexaenoic acid is a C34:6 VLCPUFA whose specific biological actions are largely unknown. This VLCPUFA, along...
Keywords: | 16Z,19Z,22Z,25Z,28Z,31Z-tetratriacontahexaenoic acid |
Application: | Bioactive Lipid Assays |
CAS | 105528-06-1 |
MW: | 496.8 D |
From 125.00€
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Item number: Cay13039-25
RD162 is a second-generation androgen receptor (AR) antagonist. It inhibits binding of 18F-FDHT to AR in human prostate cancer cells with an IC50 value of 30.9 nM. RD162 completely suppresses VCaP cell proliferation at 1 µM and induces apoptosis of VCaP cells at 10 µM. RD162 is bioavailable and reduces LNCaP/AR...
Keywords: | 4-[7-[4-cyano-3-(trifluoromethyl)phenyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methyl-benzamide |
Application: | Androgen receptor antagonist |
CAS | 915087-27-3 |
MW: | 476.4 D |
From 46.00€
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Item number: Cay13339-25
SQ 22,536 is an inhibitor of adenylyl cyclase with an IC50 value of 13 µM for inhibition of prostaglandin E1-stimulated increase in cAMP in intact platelets. It has been used to evaluate adenylyl cyclase activity during iloprost-induced vasorelaxation of isolated pulmonary veins or aorta in several research...
Keywords: | NSC 53339, 9-(tetrahydro-2-furanyl)-9H-purin-6-amine |
Application: | Adenylyl cyclase inhibitor |
CAS | 17318-31-9 |
MW: | 205.2 D |
From 84.00€
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Item number: Cay13639-25
The CXC chemokine receptor-4 (CXCR4) is a G protein-coupled receptor that is specific for stromal cell-derived factor-1 (SDF-1/ CXCL12). Activation of CXCR4 promotes homing of hematopoietic stem cells, chemotaxis and quiescence of lymphocytes, and growth and metastasis of certain cancer cell types. Moreover, CXCR4...
Keywords: | N1,N4-di-2-pyridinyl-1,4-benzenedimethanamine |
Application: | CXCR4 antagonist |
CAS | 55778-02-4 |
MW: | 290.4 D |
From 26.00€
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