4 products were found matching "Cay10162-%25"!
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GW 627368X
Item number: Cay10009162-25
The effects of prostaglandin E2 (PGE2) are transduced by at least four distinct receptors designated EP1, EP2, EP3, and EP4. GW 627368X is a potent and selective competitive antagonist of the EP4 receptor with additional human TP receptor affinity. In competition radioligand bioassays, GW 627368X had affinity for...
| Keywords: | 4-(4,9-diethoxy-1,3-dihydro-1-oxo-2H-benz[f]isoindol-2-yl)-N-(phenylsulfonyl)-benzeneacetamide |
| Application: | EP4 receptor antagonist |
| CAS | 439288-66-1 |
| MW: | 544.6 D |
From 80.00€
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15(S)-HETE Ethanolamide
Item number: Cay10169-25
Arachidonoyl ethanolamide (AEA, Cay-90050) was the first endogenous cannabinoid (CB) to be isolated and characterized as an agonist acting on the same receptors (CB1 and CB2) as THC. Since that time, a number of related endocannabinoids have been isolated, most notably 2-arachidonoyl glycerol (Cay-62160)....
| Keywords: | 15(S)-HAEA, 15(S)-hydroxy-N-(2-hydroxyethyl)-5Z,8Z,11Z,13E-eicosatetraenamide |
| Application: | Bioactive lipid assays |
| CAS | 161744-53-2 |
| MW: | 363.5 D |
From 205.00€
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Paclitaxel
Item number: Cay10461-25
Paclitaxel, a potent disruptor of microtubules derived from the bark of the Pacific yew tree, is widely used as a chemotherapeutic compound. Tested against a panel of cervical (HeLa), lung (A549), breast (MCF-7), colon (HT-29), ovarian (OVG-1), and pancreatic (PC-Sh) carcinomas, paclitaxel demonstrates IC50 values...
| Keywords: | NSC 125973, betaS-(benzoylamino)-alphaR-hydroxy-benzenepropanoic acid,... |
| Application: | Apotosis inducer |
| CAS | 33069-62-4 |
| MW: | 853.9 D |
From 43.00€
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AZD 1152-HQPA
Item number: Cay11602-25
AZD 1152-HQPA is an inhibitor of Aurora kinase B (IC50 = 0.37 nM) that demonstrates ~3,700-fold greater selectivity for Aurora kinase B over Aurora kinase A (IC50 = 1.368 µM). It does not have activity against a panel of 50 other serine-threonine or tyrosine kinases, including FLT3, JAK2, and Abl. AZD 1152-HQPA has...
| Keywords: | Barasertib-HQPA,... |
| Application: | Aurora kinase B inhibitor |
| CAS | 722544-51-6 |
| MW: | 507.6 D |
From 43.00€
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