3 products were found matching "Cay10011566-%25"!
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L-161,982
Item number: Cay10011565-25
Prostaglandin E2 (PGE2) exerts its effects through four separate G coupled-protein receptors (EP1-4). L-161,982 is a potent and selective EP4 receptor antagonist. It demonstrates selective binding to human EP4 receptors with a Ki value of 0.024 µM compared to other receptors of the prostanoid family, EP1, EP2, EP3,...
| Keywords: | N-[[4'-[[3-butyl-1,5-dihydro-5-oxo-1-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-4-yl]methyl][1,1'-biphenyl]-2-yl]sulfony... |
| Application: | EP4 receptor antagonist |
| CAS | 147776-06-5 |
| MW: | 654.7 D |
From 50.00€
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SC-51089
Item number: Cay10011561-25
SC-51089 is an antagonist of the prostaglandin E2 (PGE2) receptor subtype EP1 (Ki = 1.332 µM). It is selective for EP1 over EP2, EP3, and EP4 (Kis = >100, 17.5, and >100 µM, respectively), as well as the PGD2 receptor DP, PGF2alpha receptor FP, PGI2 receptor IP, and thromboxane A2 receptor TP (Kis = >100, 61.13,...
| Keywords: | CID132748, 8-chloro-2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide-dibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid,... |
| Application: | EP1 antagonist |
| CAS | 146033-02-5 |
| MW: | 459.3 D |
From 31.00€
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CAY10566
Item number: Cay10012562-25
Stearoyl-CoA desaturase (SCD) catalyzes the committed step of the conversion of saturated, long-chain fatty acids to monounsaturated fatty acids. The SCD1 gene is thought to play a key role in lipid homeostasis and body weight regulation. Thus, modulating SCD1 activity pharmacologically may be a useful tool for...
| Keywords: | 3-[4-(2-chloro-5-fluorophenoxy)-1-piperidinyl]-6-(5-methyl-1,3,4-oxadiazol-2-yl)-pyridazine |
| Application: | SCD inhibitor |
| CAS | 944808-88-2 |
| MW: | 389.8 D |
From 106.00€
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