3 products were found matching "Cay10011348-%25"!

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Steviol
Steviol

Item number: Cay10011344-25

Steviol is the aglycon derivative of steviol glycosides, which are natural sweeteners isolated from S. rebaudiana. Steviol inhibits human organic anion transporters (hOATs) in uptake assays using murine cells from the S2 segment of proximal tubules. It is selective for hOAT1 and hOAT3 over hOAT2 and hOAT4 (IC50s =...
Keywords: Hydroxy Dehydrostevic Acid, NSC 226902, (4alpha)-13-hydroxy-kaur-16-en-18-oic acid
Application: OAT1 / OAT3 inhibitor
CAS 471-80-7
MW: 318.5 D
From 115.00€ *
Review
Dimebolin (hydrochloride)
Dimebolin (hydrochloride)

Item number: Cay10011349-25

Dimebolin is a neuroprotective agent. It binds to histamine H1 and H2 receptors (IC50s = 3.8 and 287 nM, respectively), as well as alpha1A-, alpha1B-, alpha1D-, and alpha2A-adrenergic receptors (ARs), imidazoline I2 receptors, and the serotonin (5-HT) receptor subtypes 5-HT2A, 5-HT2C, 5-HT6, and 5-HT7 (Kis = 8-313...
Keywords: Dimebon, Latrepirdine, 2,3,4,5-tetrahydro-2,8-dimethyl-5-[2-(6-methyl-3-pyridinyl)ethyl]-1H-pyrido[4,3-b]indole,...
Application: Neuroprotective agent
CAS 97657-92-6
MW: 392.4 D
From 31.00€ *
Review
CAY10575
CAY10575

Item number: Cay10011248-25

CAY10575 inhibits IKKbeta and polo-like kinase 1 (Plk1, IC50s = 0.075 and 0.125 µM, respectively). It also inhibits IKKepsilon (IC50 = 95%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 1mg/mL, DMSO: 10mg/mL, DMSO:PBS(7.2pH) 1:4: 0.2mg/mL. lambdamax: 295 nm. SMILES:...
Keywords: 5-(5,6-dimethoxy-1H-benzimidazol-1-yl)-3-[[4-(methylsulfonyl)phenyl]methoxy]-2-thiophenecarboxamide
Application: IKKepsilon inhibitor
CAS 916985-21-2
MW: 487.6 D
From 52.00€ *
Review