3 products were found matching "Cay10010839-%25"!
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CB-13
Item number: Cay10010398-25
CB-13 is a dual agonist of the CB1 (IC50 = 15 nM) and CB2 (IC50 = 98 nM) receptors. In rats, oral CB-13 (3 mg/kg) potently blocks CB1-dependent neuropathic mechanical hyperalgesia, shows limited brain penetration, and exhibits good oral bioavailability. CB-13 does not possess genotoxic potential, as indicated by...
| Keywords: | CRA-13, 1-naphthalenyl[4-(pentylox)-1-naphthalenyl]-methanone |
| Application: | Dual CB1 / CB2 receptor agonist |
| CAS | 432047-72-8 |
| MW: | 368.5 D |
From 74.00€
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Kenpaullone
Item number: Cay10010239-25
The development of selective, cell-permeable protein kinase inhibitors for the treatment of cancer, inflammation, and other diseases, is a major focus of drug development efforts. Kenpaullone is an ATP-competitive inhibitor of several cyclin-dependent kinases (CDKs) as well as glycogen synthase kinase 3beta...
| Keywords: | 9-Bromopaullone, NSC 664704, 9-bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one |
| Application: | CDK inhibitor, GSK-3 beta inhibitor |
| CAS | 142273-20-9 |
| MW: | 327.2 D |
From 66.00€
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Lovastatin Hydroxy Acid (sodium salt)
Item number: Cay10010339-25
Lovastatin hydroxy acid is a potent and competitive inhibitor of HMG-CoA reductase (Ki = 0.6 nM). It is the more potent, open ring, hydroxy acid form of its prodrug, lovastatin (Cay-10010338).Formal Name:...
| Keywords: | 2-methyl-1S,2,3R,7S,8S,8aR-hexahydro-3,7-dimethyl-8-[2-[(2R,4R)-tetrahydro-4-hydroxy-6-oxo-2H-pyran-2-yl]ethyl]-1-naphthal... |
| Application: | NF-kappaB activation inhibitor |
| CAS | 75225-50-2 |
| MW: | 444.5 D |
From 50.00€
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