6 products were found matching "Cay10010245-%25"!

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AG-17
AG-17

Item number: Cay10010248-25

Protein tyrosine kinase (PTK) inhibitors are potential antiproliferative agents for diseases caused by the hyperactivity of protein tyrosine kinases. Tyrphostins are a class of antiproliferative compounds which act as protein tryrosine kinase blockers. PTK inhibitors which preferentially inhibit the epidermal growth...
Keywords: GCP 5126, Malonoben, NSC 242557, RG-50872, SF 6847, Tyrphostin 9, Tyrphostin AG-17,...
Application: EGF receptor kinase inhibitor
CAS 10537-47-0
MW: 282.4 D
From 38.00€ *
Review
Olomoucine
Olomoucine

Item number: Cay10010240-25

Cyclin-dependent kinases (CDKs) are key regulators of cell cycle progression and are therefore promising targets for cancer therapy. Olomoucine is a cdk inhibitor that acts by competing for the ATP binding site of the kinase. This purine derivative is an inhibitor for CDC2/cyclin B (IC50 = 7 µM), Cdk2/cyclin A (IC50...
Keywords: 2-[[9-methyl-6-[(phenylmethyl)amino]-9H-purin-2-yl]amino]-ethanol
Application: CDK inhibitor
CAS 101622-51-9
MW: 298.3 D
From 43.00€ *
Review
AG-494
AG-494

Item number: Cay10010242-25

Protein tyrosine kinase (PTK) inhibitors are potential antiproliferative agents for diseases caused by the hyperactivity of PTKs. Tyrphostins are a class of antiproliferative, compounds that act as PTK blockers. PTK inhibitors that preferentially inhibit the epidermal growth factor (EGF) receptor kinase block...
Keywords: Tyrphostin AG-494, 2E-cyano-3-(3,4-dihydroxyphenyl)-N-phenyl-2-propenamide
Application: EGF receptor kinase inhibitor
CAS 133550-35-3
MW: 280.3 D
From 46.00€ *
Review
H-8 (hydrochloride)
H-8 (hydrochloride)

Item number: Cay10010249-25

The H series isoquinolinesulfonamide protein kinase (PK) inhibitors are widely used to block signaling pathways to elucidate mechanisms of cellular regulation and signal transduction. H-8, an isoquinolinesulfonamide protein kinase (PK) inhibitor, is a potent inhibitor of PKA and PKG and shows moderate inhibition for...
Keywords: Protein Kinase Inhibitor H-8, N-[2-(methylamino)ethyl]-5-isoquinolinesulfonamide, dihydrochloride
Application: PKA inhibitor, PKG inhibitor
CAS 113276-94-1
MW: 338.3 D
From 50.00€ *
Review
AG-825
AG-825

Item number: Cay10010243-25

The HER2/Neu proto-oncogene is a member of the epidermal growth factor receptor (EGFR) family of receptor tyrosine kinases (RTK) which includes EGFR, HER2/Neu, HER3 and HER4. Overexpression of HER2/Neu occurs in 25-30% of human breast and ovarian cancer. AG-825 is a selective ATP-competitive inhibitor of the...
Keywords: Tyrphostin AG-825, 3-[3-[(2-benzothiazolylthio)methyl]-4-hydroxy-5-methoxyphenyl]-2-cyano-2-propenamide
Application: HER-2/neu inhibitor
CAS 149092-50-2
MW: 397.5 D
From 38.00€ *
Review
AG-1478
AG-1478

Item number: Cay10010244-25

Protein tyrosine kinase (PTK) inhibitors are potential antiproliferative agents for diseases caused by the hyperactivity of PTK. Tyrphostins are a class of antiproliferative compounds which act as PTK blockers. PTK inhibitors which preferentially inhibit the epidermal growth factor receptor (EGFR) kinase and block...
Keywords: NSC 693255, Tyrphostin AG-1478, N-(3-chlorophenyl)-6,7-dimethoxy-4-quinazolinamine
Application: EGF receptor kinase inhibitor
CAS 153436-53-4
MW: 315.8 D
From 30.00€ *
Review