3 products were found matching "Cay10010182-%25"!
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AM1241
Item number: Cay10010118-25
AM1241 is a cannabinoid (CB) receptor agonist that is selective for CB2 over CB1 with Ki values of 7.1 and 580 nM for human recombinant receptors transfected into HEK and CHO cells, respectively, in a radioligand binding assay. It is considered a protean agonist as it has neutral antagonist and partial agonist...
| Keywords: | (2-iodo-5-nitrophenyl)-(1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl)methanone |
| Application: | CB2 receptor agonist |
| CAS | 444912-48-5 |
| MW: | 503.3 D |
From 43.00€
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(R)-Equol
Item number: Cay10010172-25
(R)-Equol is an agonist of estrogen receptor alpha (ERalpha) and active metabolite of the polyketide isoflavone daidzein (Cay-10005166). It is formed from daidzein by gut microbiota. (R)-Equol selectively induces ERalpha-mediated gene transcription over ERbeta-mediated transcription in HEC-1 cells expressing the...
| Keywords: | (+)-Equol, Isoequol, 3,4-dihydro-3R-(4-hydroxyphenyl)-2H-1-benzopyran-7-ol |
| Application: | ERalpha agonist |
| CAS | 221054-79-1 |
| MW: | 242.3 D |
From 24.00€
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PD 146176
Item number: Cay10010518-25
PD 146176 is a potent and selective inhibitor of reticulocyte 15-lipoxygenase-1. It limits hypercholesterolemia-induced atherosclerosis in New Zealand White rabbits and reduces oxidant stress-induced apoptosis in endothelial cells. PD 146176 inhibits amyloid beta protein aggregate formation without changing total...
| Keywords: | NSC 168807, 6,11-dihydro-[1]benzothiopyrano[4,3-b]indole |
| Application: | 15-LO inhibitor |
| CAS | 4079-26-9 |
| MW: | 237.3 D |
From 65.00€
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