6 products were found matching "Cay10005368-%25"!
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1,2-Dioleoyl-rac-glycerol
Item number: Cay10007863-25
1,2-Dioleoyl-rac-glycerol is a diacylglycerol that contains oleic acid at the sn-1 and sn-2 positions. It effectively binds the C1 domain to activate conventional protein kinase C forms and serves as a substrate for DAG kinases and multisubstrate lipid kinase.Formal Name: 9Z-octadecenoic acid,...
| Keywords: | (±)-1,2-Diolein, rac-Glycerol 1,2-dioleate, 9Z-octadecenoic acid, 1,1'-[1-(hydroxymethyl)-1,2-ethanediyl] ester |
| Application: | PKC activator, kinase substrate |
| CAS | 2442-61-7 |
| MW: | 621 D |
From 60.00€
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CAY10508
Item number: Cay10008669-25
Central cannabinoid (CB1) receptor antagonists and inverse agonists exhibit therapeutic potential for obesity and drug dependence, while being devoid of psychotropic effects. CAY10508 is a potent and selective central cannabinoid (CB1) receptor inverse agonist with a Ki value of 243 nM and an EC50 of 195 nM. A 10 µM...
| Keywords: | 1,3-bis(4-bromophenyl)-5-phenyl-2,4-imidazolidinedione |
| Application: | CB1 receptor inverse agonist |
| CAS | 878533-35-8 |
| MW: | 486.2 D |
From 38.00€
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O-1602
Item number: Cay10006803-25
O-1602 (Cay-10006803) is an analytical reference standard that is structurally similar to known phytocannabinoids. O-1602 has been found in Cannabis. This product is intended for research and forensic applications.Formal Name: 5-methyl-4-[(1R,6R)-3-methyl-6-(1-methylethenyl)-2-cyclohexen-1-yl]-1,3-benzenediol. CAS...
| Keywords: | Abn-CBDO, Abnormal Cannabidiorcin, Abnormal Cannabidiorcinol, Abnormal Cannabiorcodiol,... |
| Application: | Cannabidiol analog |
| CAS | 317321-41-8 |
| MW: | 258.4 D |
From 39.00€
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GW 5074
Item number: Cay10010368-25
Raf-1 is a proto-oncogene serine/threonine protein kinase that signals from Ras to the MAPK/ERK signaling pathway. This pathway mediates basic cellular functions, including proliferation, differentiation, and survival. GW 5074 is a potent, selective, and cell-permeable inhibitor of Raf-1 (IC50 = 9 nM). It blocks...
| Keywords: | 3-[(3,5-dibromo-4-hydroxyphenyl)methylene]-1,3-dihydro-5-iodo-2H-indol-2-one |
| Application: | Raf-1 inhbitor |
| CAS | 220904-83-6 |
| MW: | 520.9 D |
From 50.00€
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Exemestane
Item number: Cay15008-25
Exemestane is an irreversible inhibitor of aromatase (Ki = 26 nM). It is selective for aromatase over 5alpha-reductase when used at a concentration of 30 µM. Subcutaneous administration of exemestane (3-100 mg/kg per day) decreases tumor proliferation in rats with mammary tumors induced by the carcinogenic...
| Keywords: | Aromasin(TM), FCE 24304, 6-methylene-androsta-1,4-diene-3,17-dione |
| Application: | Steroidal aromatase inhibitor |
| CAS | 107868-30-4 |
| MW: | 296.4 D |
From 60.00€
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Trifluoperazine (hydrochloride)
Item number: Cay15068-25
Trifluoperazine (TFP) is a phenothiazine compound with anti-adrenergic and anti-dopaminergic actions typical of antipsychotic agents. It antagonizes adrenergic receptors, with selectivity for alpha1 over the alpha2 subtypes (Kis = 24, 653, 163, and 391 nM for alpha1A, alpha2A, alpha2B, and alpha2C, respectively)....
| Keywords: | SKF 5019, TFP, 10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoromethyl)-10H-phenothiazine, dihydrochloride |
| Application: | Dopamine receptor D2 antagonist |
| CAS | 440-17-5 |
| MW: | 480.4 D |
From 43.00€
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