9 products were found matching "Cay10003-%25"!

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Lipoxin A4 methyl ester
Lipoxin A4 methyl ester

Item number: Cay10033-25

Lipoxin A4 (LXA4) methyl ester is a more lipid soluble, prodrug formulation of the transcellular metabolite LXA4. LXA4 is a trihydroxy fatty acid containing a conjugated tetraene, produced by the metabolism of 15-HETE or 15-HpETE with human leukocytes. LXA4 is equipotent to leukotriene B4 (LTB4) in inducing...
Keywords: 5(S),6(R),15(S)-TriHETE methyl ester, LXA4 methyl ester, 5S,6R,15S-trihydroxy-7E,9E,11Z,13E-eicosatetraenoic acid, methyl...
Application: Bioactive lipid assays
CAS 97643-35-1
MW: 366.5 D
From 368.00€ *
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G-1
G-1

Item number: Cay10008933-25

GPR30 is a transmembrane G protein-coupled receptor (GPCR) localized to endoplasmic reticulum (ER) that binds estradiol with high affinity, activating multiple intracellular signaling pathways. G-1 is a nonsteroidal, high-affinity, selective agonist of GPR30 that binds with a Ki value of 11 nM. Competitive binding...
Keywords: rel-1-[4-(6-bromo-1,3-benzodioxol-5-yl)-3aR,4S,5,9bS-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]-ethanone
Application: GPR30 agonist
CAS 881639-98-1
MW: 412.3 D
From 44.00€ *
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Prostaglandin F2alpha-d9
Prostaglandin F2alpha-d9

Item number: Cay10008643-25

Prostaglandin F2alpha-d9 (PGF2alpha-d9) contains nine deuterium atoms at the 17, 17', 18, 18', 19, 19', 20, 20, and 20 positions. It is intended for use as an internal standard for the quantification of PGF2alpha by GC- or LC-mass spectrometry. PGF2alpha is a widely distributed PG occurring in many species. It...
Keywords: Dinoprost-d9, 9alpha,11alpha,15S-trihydroxy-prosta-5Z,13E-dien-1-oic-17,17,18,18,19,19,20,20,20-d9 acid
Application: Standard
MW: 363.5 D
From 65.00€ *
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3-thio-Pheneacrylic Acid
3-thio-Pheneacrylic Acid

Item number: Cay10007103-25

3-thio-Pheneacrylic acid is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 3-(3-thienyl)-2-propenoic acid. CAS Number: 1195-52-4. Synonyms: 3-Thiophen-3-yl-Acrylic Acid. Molecular Formula: C7H6O2S. Formula Weight: 154.2. Purity: >98%. Formulation: (Request formulation change), A...
Keywords: 3-Thiophen-3-yl-Acrylic Acid, 3-(3-thienyl)-2-propenoic acid
Application: Synthetic intermediate, Pharmaceutical synthesis
CAS 1195-52-4
MW: 154.2 D
From 26.00€ *
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1,2-Dioleoyl-rac-glycerol
1,2-Dioleoyl-rac-glycerol

Item number: Cay10007863-25

1,2-Dioleoyl-rac-glycerol is a diacylglycerol that contains oleic acid at the sn-1 and sn-2 positions. It effectively binds the C1 domain to activate conventional protein kinase C forms and serves as a substrate for DAG kinases and multisubstrate lipid kinase.Formal Name: 9Z-octadecenoic acid,...
Keywords: (±)-1,2-Diolein, rac-Glycerol 1,2-dioleate, 9Z-octadecenoic acid, 1,1'-[1-(hydroxymethyl)-1,2-ethanediyl] ester
Application: PKC activator, kinase substrate
CAS 2442-61-7
MW: 621 D
From 60.00€ *
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2-Aminopyrazine
2-Aminopyrazine

Item number: Cay10007093-25

2-Aminopyrazine is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: pyrazinamine. CAS Number: 5049-61-6. Synonyms: NSC 13147. Molecular Formula: C4H5N3. Formula Weight: 95.1. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 20 mg/ml, DMSO: 20...
Keywords: NSC 13147, pyrazinamine
Application: Synthetic intermediate, Pharmaceutical synthesis
CAS 5049-61-6
MW: 95.1 D
From 26.00€ *
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HMB-Val-Ser-Leu-VE
HMB-Val-Ser-Leu-VE

Item number: Cay10007713-25

HMB-Val-Ser-Leu-VE is a cell-permeable vinyl ester tripeptide inhibitor of the trypsin-like activity of the 20S proteasome (IC50 = 0.033 µM). It is selective for the trypsin-like activity over the chymotryptic- or post-acidic-like activities (IC50s = >10 µM for both). HMB-Val-Ser-Leu-VE is active against T. brucei...
Keywords: N-(3-hydroxy-2-methylbenzoyl)-L-valyl-N-[(1S,2E)-4-ethoxy-1-(2-methylpropyl)-4-oxo-2-butenyl]-L-serinamide
Application: 20S proteasome inhibitor
CAS 862891-04-1
MW: 505.6 D
From 96.00€ *
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PSN375963
PSN375963

Item number: Cay10008593-25

GPR119 (previously designated SNORF25) is an orphan G protein-coupled receptor expressed predominantly in the pancreas and gastrointestinal tract in humans and in the brain, pancreas, and gastrointestinal tract in rodents. It mediates a reduction in food intake and body weight gain in rats upon treatment with oleoyl...
Keywords: 4-[5-(4-butylcyclohexyl)-1,2,4-oxadiazol-3-yl]-pyridine
Application: GPR119 agonist
CAS 388575-52-8
MW: 285.4 D
From 24.00€ *
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CAY10734
CAY10734

Item number: Cay10007833-25

CAY10734 is an agonist of sphingosine-1-phosphate receptor 1 (S1P1, IC50 = 0.6 nM). It selectively binds S1P1 over S1P2, S1P3, and S1P4 receptors (IC50s = >10,000, 12,000, and 70 nM, respectively) but does also bind S1P5 receptors (IC50 = 1 nM) in radioligand binding assays. CAY10734 reduces the number of peripheral...
Keywords: 1-[[4-[5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]methyl]-3-azetidinecarboxylic acid
Application: S1P1 receptor agonist
CAS 635701-59-6
MW: 391.5 D
From 43.00€ *
Review