5 products were found matching "Cay100017-%25"!
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HMB-Val-Ser-Leu-VE
Item number: Cay10007713-25
HMB-Val-Ser-Leu-VE is a cell-permeable vinyl ester tripeptide inhibitor of the trypsin-like activity of the 20S proteasome (IC50 = 0.033 µM). It is selective for the trypsin-like activity over the chymotryptic- or post-acidic-like activities (IC50s = >10 µM for both). HMB-Val-Ser-Leu-VE is active against T. brucei...
| Keywords: | N-(3-hydroxy-2-methylbenzoyl)-L-valyl-N-[(1S,2E)-4-ethoxy-1-(2-methylpropyl)-4-oxo-2-butenyl]-L-serinamide |
| Application: | 20S proteasome inhibitor |
| CAS | 862891-04-1 |
| MW: | 505.6 D |
From 96.00€
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Renin (human, recombinant)
Item number: Cay10006217-25
Renin is an aspartyl protease glycoprotein, a member of the aspartic acid protease family, and a hormone. It is a single-chain polypeptide in which the N- and C-terminal portions contain an aspartate residue responsible for its catalytic activity. It is formed from prorenin, a zymogen found primarily in the...
| Keywords: | REN, Renin, Renin, Angiotensinogenase, Angiotensinogenase |
| Application: | Enzyme activity, WB |
514.00€
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PAC-1
Item number: Cay10009317-25
Apoptosis can be induced when procaspase-3 is activated and converted to caspase-3. Procaspase-activating compound 1 (PAC-1) is a procaspase-3 activator and a potential drug treatment in cancer cell lines with elevated levels of procaspase-3. PAC-1's effectiveness was found to be directly proportional to the...
| Keywords: | Procaspase-activating Compound 1, 4-(phenylmethyl)-1-piperazineacetic acid,... |
| Application: | Procaspase-3 activator |
| CAS | 315183-21-2 |
| MW: | 392.5 D |
From 145.00€
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Arachidonic Acid Leelamide
Item number: Cay10008617-25
Arachidonic acid leelamide is the arachidonic amide analog of leelamine. Leelamine has weak affinity for the human central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 µM. Leelamine inhibits pyruvate dehydrogenase kinase (PDK) with...
| Keywords: | 1R,2,3,4,4aS,9,10,10aR-octahydro-1,4a-dimethyl-7-(1-methylethyl)-1-phenanthrene-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Application: | Bioactive lipid assays |
| MW: | 571.9 D |
From 72.00€
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PtdIns-(3,4,5)-P3 Binding Protein
Item number: Cay10009817-25
Pleckstrin homology (PH) domains all contain a seven-standard beta-sandwich that allows binding to various species of phosphatidyl inositol (PtdIns) phosphates. Most PH domains bind to PtdIns phosphates with weak affinity and low specificity. However, a small subclass binds specifically and with high-affinity for...
| Keywords: | Grp1, Grp1, ARNO3, Cytohesin-3, Cytohesin-3, Protein ARNO3, Protein ARNO3, ARF nucleotide-binding site opener 3, ARF... |
| Application: | WB |
| MW: | 41,7 kD |
From 189.00€
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