3 products were found matching "Cay70705"!
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U-75302
Item number: Cay70705-100
U-75302 is an LTB4 receptor antagonist with a Ki of 159 nM on guinea pig lung membranes. This activity is specific for the BLT1 receptor, U-75302 does not antagonize the binding of [3H]-LTB4 to the human BLT2 receptor.Formal Name: 6-(6-(3R-hydroxy-1E,5Z-undecadien-1-yl)-2-pyridinyl)-1,5S-hexanediol. CAS Number:...
| Keywords: | 6-(6-(3R-hydroxy-1E,5Z-undecadien-1-yl)-2-pyridinyl)-1,5S-hexanediol |
| Application: | LTB4 receptor antagonist |
| CAS | 119477-85-9 |
| MW: | 361.5 D |
From 117.00€
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Bromoenol lactone
Item number: Cay70700-5
BEL is a selective, potent, irreversible, mechanism-based inhibitor of myocardial cytosolic calcium-independent phospholipase A2 (iPLA2) with a Ki value of 180 nM. BEL also inhibits macrophage iPLA2 in a concentration-dependent manner with an IC50 value of 60 nM and is an effective enzyme-activated irreversible...
| Keywords: | BEL, Haloenol lactone, HELSS, 6E-(bromomethylene)tetrahydro-3-(1-naphthalenyl)-2H-pyran-2-one |
| Application: | iPLA2 inhibitor |
| CAS | 88070-98-8 |
| MW: | 317.2 D |
From 161.00€
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U-73122
Item number: Cay70740-5
U-73122 is an inhibitor of PLC-dependent processes, however, the mechanism of action remains unclear. The IC50 values for inhibition of platelet aggregation induced by collagen or thrombin are 0.6 and 5 µM, respectively. It also exhibits inhibitory activity against HIV-1 integrase with an IC50 value of 7 µM.Formal...
| Keywords: | 1-[6-[[(17beta)-3-methoxyestra-1,3,5(10)-trien-17-yl]amino]hexyl]-1H-pyrrole-2,5-dione |
| Application: | Lipid signaling studies |
| CAS | 112648-68-7 |
| MW: | 464.6 D |
From 28.00€
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