- Search results for Cay15773
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3 products were found matching "Cay15773"!
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Item number: Cay15773-5
Tiotropium is an antagonist that binds to M1, M2, and M3 muscarinic acetylcholine receptors (Kds = 0.43, 0.54, and 0.69 nM, respectively, for human receptors). It decreases acetylcholine-induced contraction of isolated guinea pig trachea in a concentration-dependent manner. In vivo, tiotropium (1 g/L inhaled...
Keywords: | BA 679BR,... |
Application: | Muscarinic cholinergic receptor antagonist |
CAS | 136310-93-5 |
MW: | 472.4 D |
From 98.00€
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Item number: Cay11573-10
IOX2 is an inhibitor of hypoxia-inducible factor prolyl hydroxylase 2 (HIF-PH2, IC50 = 21 nM) with over 100-fold selectivity compared to inhibition of JMJD2A, JMJD2C, JMJD2E, JMJD3, or the 2OG oxygenase FIH (IC50s > 100 µM). IOX2 is active in cells, inhibiting HIF-1alpha hydroxylation in RCC4 cells at 50 µM. See the...
Keywords: | N-[[1,2-dihydro-4-hydroxy-2-oxo-1-(phenylmethyl)-3-quinolinyl]carbonyl]-glycine |
Application: | PHD2 inhibitor |
CAS | 931398-72-0 |
MW: | 352.3 D |
From 92.00€
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Item number: Cay15573-10
Inactivation of the tumor suppressor p53 commonly coincides with increased signaling through NF-kappaB in cancer. CAY10681 is a dual modulator of p53-MDM2 interaction and NF-kappaB signaling. It potently binds MDM2 (Ki = 250 nM), reducing MDM2-mediated turnover of p53. CAY10681 also inhibits phosphorylation of...
Keywords: | 4-(4-bromophenyl)-4,5-dihydro-5-[3-(1H-imidazol-1-yl)propyl]-3-phenyl-1-(phenylmethyl)-pyrrolo[3,4-c]pyrazol-6(1H)-one |
Application: | p53-MDM2 interaction / NF-kappaB signaling modulator |
CAS | 1542066-69-2 |
MW: | 552.5 D |
From 98.00€
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