- Search results for Cay14400
Cookie preferences
This website uses cookies, which are necessary for the technical operation of the website and are always set. Other cookies, which increase the comfort when using this website, are used for direct advertising or to facilitate interaction with other websites and social networks, are only set with your consent.
Configuration
Technically required
These cookies are necessary for the basic functions of the shop.
"Allow all cookies" cookie
"Decline all cookies" cookie
CSRF token
Cookie preferences
Currency change
Customer-specific caching
FACT-Finder tracking
Individual prices
Selected shop
Session
Comfort functions
These cookies are used to make the shopping experience even more appealing, for example for the recognition of the visitor.
Note
Show the facebook fanpage in the right blod sidebar
Statistics & Tracking
Affiliate program
Conversion and usertracking via Google Tag Manager
Track device being used
17 products were found matching "Cay14400"!
Close filters
Filter by:
No results were found for the filter!
Item number: Cay14400-1
Thioridazine is a typical antipsychotic. It binds to dopamine D2, histamine H1, M3 muscarinic, and alpha1- and alpha2-adrenergic receptors (Kis = 5-341.3 nM), as well as the serotonin (5-HT) receptor subtypes 5-HT1A, 5-HT2A, 5-HT2C, 5-HT6, and 5-HT7 (Kis = 10-180.7 nM). Thioridazine (5 mg/kg) reduces...
Keywords: | Aldazine, NSC 186060, 10-[2-(1-methyl-2-piperidinyl)ethyl]-2-(methylthio)-10H-phenothiazine, monohydrochloride |
Application: | Dopamine D2-receptor antagonist |
CAS | 130-61-0 |
MW: | 407 D |
From 43.00€
*
Item number: Cay11440-5
Gram negative bacteria utilize N-acylated homoserine lactones to coordinate expression of virulence in response to the density of the surrounding bacterial population in a process termed quorum sensing. By interfering with this communication and thereby disrupting virulence expression, quorum sensing inhibitors are...
Keywords: | NSC 402844, 3-methoxy-5-methyl-4-oxo-2,5-hexadienoic acid |
Application: | Antibiotic |
CAS | 90-65-3 |
MW: | 170.2 D |
From 66.00€
*
Item number: Cay14440-5
The poly(ADP-ribose) polymerases (PARPs) form a family of enzymes with roles in DNA repair and apoptosis, particularly in response to reactive oxygen and nitrogen species. PJ-34 is an inhibitor of PARPs which can be used in cells or in animals. It binds and inhibits the PARP tankyrase1 (IC50 = 1 µM). PJ-34 also...
Keywords: | N-(5,6-dihydro-6-oxo-2-phenanthridinyl)-2-(dimethylamino)-acetamide, monohydrochloride |
Application: | PARP inhibitor |
CAS | 344458-15-7 |
MW: | 331.8 D |
From 50.00€
*
Item number: Cay14000-25
Auraptene is a coumarin derived from citrus plants that bears a geranyloxyl moiety at its C-7. It has anti-inflammatory, anti-carcinogenic, anti-bacterial, neuroprotective, and hepatoprotective activities. It inhibits leukocyte activation and induces phase II enzymes during the initiation phase of carcinogenesis....
Keywords: | 7-Geranyloxycoumarin, 7-[[(2E)-3,7-dimethyl-2,6-octadien-1-yl]oxy]-2H-1-benzopyran-2-one |
Application: | Metabolic studies |
CAS | 495-02-3 |
MW: | 298.4 D |
From 39.00€
*
Item number: Cay11140-10
The NF-kappaB/Rel family of transcription factors induce and coordinate the expression of pro-inflammatory genes including cytokines, chemokines, interferons, MHC proteins, growth factors, and cell adhesion molecules. Under resting conditions NF-kappaB dimers are retained in the cytoplasm by a member of the IkappaB...
Keywords: | 3-[(aminocarbonyl)amino]-5-[4-(4-morpholinylmethyl)phenyl]-2-thiophenecarboxamide |
Application: | Potential IKK-2 inhibitor |
CAS | 494772-86-0 |
MW: | 360.4 D |
From 58.00€
*
Item number: Cay14405-50
Glycerophosphate is a mixture of the endogenous metabolite alpha-glycerophosphate and the alkaline phosphatase (ALP) inhibitor beta-glycerophosphate (Cay-38367).Formal Name: 1,2,3-propanetriol, 2-(dihydrogen phosphate), 1,2,3-propanetriol, (2R)1-(dihydrogen phosphate), disodium salt, pentahydrate. Synonyms: Glycerol...
Keywords: | 2-(dihydrogen phosphate)-1,2,3-propanetriol, disodium salt, pentahydrate |
Application: | Protein phosphatase inhibitor |
MW: | 306.1 D |
From 66.00€
*
Item number: Cay14406-10
Sodium-hydrogen exchangers (NHE) are involved in maintaining sodium and pH balance in a variety of tissues. They are also known as sodium-hydrogen antiporters and solute carrier family 9 members. 5-(N-ethyl-N-isopropyl)-Amiloride (EIPA) is a potent inhibitor of several NHE isoforms, inhibiting NHE1, NHE2, NHE3, and...
Keywords: | EIPA, L-593,754, MH 12-43, 3-amino-N-(aminoiminomethyl)-6-chloro-5-[ethyl(1-methylethyl)amino]-2-pyrazinecarboxamide |
Application: | NHE inhibitor |
CAS | 1154-25-2 |
MW: | 299.8 D |
From 77.00€
*
Item number: Cay14408-50
Bucladesine is a cell-permeable, cyclic nucleotide derivative that mimics the action of endogenous cyclic adenosine monophosphate (cAMP) and is a phosphodiesterase inhibitor. Because it mimics cAMP and can induce normal physiological responses when added to cells in experimental conditions, bucladesine is widely...
Keywords: | DC 2797, N-(1-oxobutyl)-cyclic 3',5'-(hydrogen phosphate) 2'-butanoate-adenosine, monosodium salt |
Application: | Cell-permeable cAMP mimic |
CAS | 16980-89-5 |
MW: | 491.4 D |
From 48.00€
*
Item number: Cay14407-10
SIRT1/2 inhibitor IV is a cell-permeable inhibitor of SIRT1 (IC50 = 56 µM) and SIRT2 (IC50 = 59 µM), blocking NAD+-dependent deacetylase activity in a substrate competitive manner. It less effectively inhibits SIRT5 (IC50 >300 µM) and has no effect on class I and II histone deacetylases. By inhibiting SIRT1, SIRT1/2...
Keywords: | Cambinol, NSC 112546, SIRT1 Inhibitor II, SIRT2 Inhibitor VI,... |
Application: | SIRT1/2 inhibitor |
CAS | 14513-15-6 |
MW: | 360.4 D |
From 43.00€
*
Item number: Cay14404-10
A-771726 is an active metabolite of the prodrug leflunomide (Cay-14860) that inhibits dihydroorotate dehydrogenase (DHODH, IC50 = 0.23 µM). A-771726 inhibits the production of prostaglandin E2 (PGE2, Cay-14010) in TNF-alpha- or IL-1alpha-stimulated isolated human synoviocytes (IC50s = 7 and 3 µM, respectively). It...
Keywords: | Flucyamide, HMR 1726, SU 20, Teriflunomide, 2-cyano-3-hydroxy-N-[4-(trifluoromethyl)phenyl]-2Z-butenamide |
Application: | Dihydroorotate dehydrogenase inhibitor, Tyrosine kinase inhibitor |
CAS | 163451-81-8 |
MW: | 270.2 D |
From 84.00€
*
Item number: Cay14423-100
Rifampicin is a rifamycin antibiotic and inhibitor of bacterial RNA polymerase (IC50 = 0.01 µg/ml for the E. coli enzyme). It inhibits the growth of M. tuberculosis H37Rv in mouse peritoneal macrophages (MIC = 0.8 µg/ml) as well as clinical isolates of various species of Staphylococcus, Streptococcus, Haemophilus,...
Keywords: | NIH 10782, NSC 113926, Rifampin, 3-[[(4-methyl-1-piperazinyl)imino]methyl]-rifamycin |
Application: | Antibacterial Agent |
CAS | 13292-46-1 |
MW: | 823 D |
From 43.00€
*
Item number: Cay14429-500
AM2201 N-(3-chloropentyl) isomer is a synthetic cannabinoid which differs from AM2201 by having a 3-chloro group rather than a 5-fluoro group on the pentyl chain. The physiological and toxicological properties of this compound are not established. This product is for forensic and research applications.Formal Name:...
Keywords: | AM2201 N-(3-chloropentyl) analog, 1-(5-fluoropentyl)-1H-indole-3-carboxylic acid, 3-quinolinyl ester |
Application: | Analytical reference standard, Synthetic cannabinoid analog |
CAS | 2365471-18-5 |
MW: | 375.9 D |
From 235.00€
*