3 products were found matching "Cay14495-100"!

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HA-100 (hydrochloride)
HA-100 (hydrochloride)

Item number: Cay14955-10

HA-100 is an isoquinoline compound with an added piperazinylsulfonyl group that acts as an inhibitor of protein kinases (PKs), including PKA, PKC, and PKG (IC50s = 8, 12, and 4 µM, respectively). It less effectively blocks the activity of myosin light chain kinase (IC50 = 240 µM).Formal Name:...
Keywords: C-1, 5-(1-piperazinylsulfonyl)-isoquinoline, dihydrochloride
Application: Protein kinase inhbitor
CAS 210297-47-5
MW: 350.3 D
From 85.00€ *
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Cediranib
Cediranib

Item number: Cay11495-10

Receptors for VEGF have central roles in vasculogenesis and angiogenesis and thus serve as targets for cancer therapy. Cediranib is a potent inhibitor of VEGF receptor tyrosine kinases, including VEGFR1, 2, and 3 (IC50s = 5, 1, and 3 nM, respectively). It also potently inhibits a variety of other receptor and...
Keywords: AZD 2171, ZD 2171, 4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]-quinazoline
Application: VEGFR1/2/3 inhibitor
CAS 288383-20-0
MW: 450.5 D
From 119.00€ *
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17-trans Prostaglandin E3
17-trans Prostaglandin E3

Item number: Cay14995-100

17-trans Prostaglandin E3 (17-trans PGE3) is an isomer of PGE3 which could theoretically result from the COX metabolism of dietary trans-fatty acids. There are no published reports on the biological activity of this compound.Formal Name: 11alpha,15S-dihydroxy-9-oxo-prosta-5Z,13E,17E-trien-1-oic acid. CAS Number:...
Keywords: 17-trans PGE3, 9-oxo-11alpha,15S-dihydroxy-prosta-5Z,13E,17E-trien-1-oic acid
Application: Bioactive lipid assays
CAS 210979-33-2
MW: 350.5 D
From 115.00€ *
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