2 products were found matching "Cay15752"!

No results were found for the filter!
CFTR Inhibitor II
CFTR Inhibitor II

Item number: Cay15772-50

The cystic fibrosis (CF) gene encodes a cAMP-regulated chloride channel, the CF transmembrane conductance regulator (CFTR). CFTR inhibitor II, also known as GlyH-101, is a glycine hydrazide that selectively and reversibly blocks the CFTR channel (Ki = 4.3 µM). This compound binds to a site at the external pore of...
Keywords: Cystic Fibrosis Transmembrane Conductance Regulator Inhibitor II, GlyH-101,...
Application: CF transmembrane conductance regulator inhibitor
CAS 328541-79-3
MW: 493.2 D
From 56.00€ *
Review
Bufalin
Bufalin

Item number: Cay15725-5

Bufalin is a cardiotonic steroid first isolated from toad venom and used in traditional Asian medicine. It inhibits the Na+/K+-ATPase transporter (Kds = 42, 45, and 40 nM for the alpha1, alpha2, and alpha3 subunits, respectively). Intravenously administered bufalin is cleared rapidly, with a plasma half-life of 25...
Keywords: NSC 89595, (3beta,5beta)-3,14-dihydroxy-bufa-20,22-dienolide
Application: Na+/K+-ATPase transporter inhibitor, SRC-1/3 inhibitor
CAS 465-21-4
MW: 386.5 D
From 77.00€ *
Review