3 products were found matching "Cay70255-0.1"!

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(±)-Flurbiprofen
(±)-Flurbiprofen

Item number: Cay70250-1000

(±)-Flurbiprofen is a non-selective COX inhibitor (IC50s = 0.04 and 0.51 µM for COX-1 and COX-2, respectively). In vivo, (±)-flurbiprofen (0.3-4.8 mg/kg, p.o.) reduces carrageenan-induced hind paw edema and yeast-induced fever in rats. (±)-Flurbiprofen reduces plasma fibrinogen levels and arthritic score in a rat...
Keywords: Ansaid, (±)-2-fluoro-alpha-methyl-[1,1'-biphenyl]-4-acetic acid
Application: COX inhibitor
CAS 5104-49-4
MW: 244.3 D
From 43.00€ *
Review
(R)-Flurbiprofen
(R)-Flurbiprofen

Item number: Cay70255-1

(R)-Flurbiprofen is a COX-inactive enantiomer of the racemic non-selective COX inhibitor flurbiprofen (Cay-70250) that has diverse biological activities. It inhibits gamma-secretase activity in vitro and, in vivo, it reduces formation of amyloid-beta peptide 1-42 (Abeta42) and improves axonal transport in young...
Keywords: E-7869, Flurizan, Tarenflurbil, (R)-(-)-2-fluoro-alpha-methyl-4-biphenylacetic acid
Application: Gamma secretase inhibitor
CAS 51543-40-9
MW: 244.3 D
From 43.00€ *
Review
IMMA
IMMA

Item number: Cay70275-50

IMMA is a cannabinoid (CB) receptor 2 inverse agonist (Ki = 435 nM for recombinant human CB2). It is selective for CB2 over CB1 receptors (Ki = >20 µM). IMMA (0.001-1 µM) reduces basal production of inositol phosphate and increases forskolin-induced accumulation of cAMP in HEK293 cells expressing human CB2...
Keywords: BML-190, Indomethacin Morpholinylamide, LM-4131,...
Application: CB2 receptor agonist
CAS 2854-32-2
MW: 426.9 D
From 35.00€ *
Review