6 products were found matching "Cay9000655-50"!

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(±)-2-Methyl Arachidonoyl-2'-Fluoroethylamide
(±)-2-Methyl Arachidonoyl-2'-Fluoroethylamide

Item number: Cay90055-50

(±)-2-Methyl arachidonoyl-2'-fluoroethylamide (2-Methyl-2'-fluoro AEA) is an analog of anandamide (AEA) in which the alcohol of the ethanolamide group has been removed and replaced with a fluorine atom. This substitution confers considerably increased binding affinity for the CB1 receptor (Ki = 5.7 nM in rat brain)....
Keywords: 2-methyl-2'-fluoro AEA, 2-Methyl-2'-fluoro Anandamide, O-689, (±)-N-(2-fluoroethyl)-2-methyl-5Z,8Z,11Z,14Z-eicosatetraenamide
Application: FAAH substrate
CAS 166100-39-6
MW: 363.6 D
From 34.00€ *
Review
Dimebolin
Dimebolin

Item number: Cay9000556-5

Dimebolin is a neuroprotective agent. It binds to histamine H1 and H2 receptors (IC50s = 3.8 and 287 nM, respectively), as well as alpha1A-, alpha1B-, alpha1D-, and alpha2A-adrenergic receptors (ARs), imidazoline I2 receptors, and the serotonin (5-HT) receptor subtypes 5-HT2A, 5-HT2C, 5-HT6, and 5-HT7 (Kis = 8-313...
Keywords: Dimebon(TM), Latrepirdine, 2,3,4,5-tetrahydro-2,8-dimethyl-5-[2-(6-methyl-3-pyridinyl)ethyl]-1H-pyrido[4,3-b]indole
Application: Neuroprotective agent
CAS 3613-73-8
MW: 319.4 D
From 28.00€ *
Review
Progesterone 3-PEG11-biotin
Progesterone 3-PEG11-biotin

Item number: Cay9000645-500

Progesterone, along with pregnenolone, is the biosynthetic precursor of all other steroid hormones. Progesterone is synthesized from cholesterol by the sequential action of desmolase in the mitochondria, which produces pregnenolone, followed by Delta4,5-isomerase in the outer mitochondrial membrane and smooth...
Keywords: N-(1-(((E)-(17-acetyl-10,13-dimethyl-7,8,9,11,12,13,14,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-3(2H,6H,10H)-ylidene...
Application: Affinity probe (progesterone detection)
MW: 1140.5 D
From 125.00€ *
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Latanoprost-d4
Latanoprost-d4

Item number: Cay10006556-50

Latanoprost-d4 is intended for use as an internal standard for the quantification of latanoprost (Cay-16812) by GC- or LC-MS. Latanoprost is a derivative of prostaglandin F2alpha (PGF2alpha, Cay-16010, Cay-16020), an FP receptor agonist, and a prodrug of latanoprost (free acid) (Cay-16811). It induces...
Keywords: 17-phenyl-13,14-dihydro trinor Prostaglandin F2alpha-d4 isopropyl ester,...
Application: Standard
MW: 436.6 D
From 60.00€ *
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CAY10464
CAY10464

Item number: Cay10006545-50

The aryl hydrocarbon receptor (AhR) is a ligand-dependent intracellular transcription factor whose ligands include some of the most infamous xenobiotics, including dioxin (TCDD, 2,3,7,8-tetrachlorodibenzoparadioxin), benzo[a]pyrene, and numerous polyaromatic hydrocarbons from soot particles and coal tar. CAY10464 is...
Keywords: 1,3-dichloro-5-[(1E)-2-(4-methoxyphenyl)ethenyl]-benzene
Application: AhR antagonist
CAS 688348-37-0
MW: 279.2 D
From 30.00€ *
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Arachidonoyl Ethanolamide
Arachidonoyl Ethanolamide

Item number: Cay90050-50

Arachidonoyl ethanolamide (AEA) is the ethanolamine amide of arachidonic acid, originally isolated from porcine brain. AEA is an endogenous cannabinoid neurotransmitter that binds to both cannabinoid 1 (CB1) and CB2 receptors. AEA has Ki values ranging from 61 to 543 nM for CB1 receptors and from 279 to 1,940 nM for...
Keywords: AEA, Anandamide, N-(2-hydroxyethyl)-5Z,8Z,11Z,14Z-eicosatetraenamide
Application: Bioactive Lipid assays
CAS 94421-68-8
MW: 347.5 D
From 54.00€ *
Review