4 products were found matching "Cay16478-50"!
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Promethazine (hydrochloride)
Item number: Cay16478-10
Promethazine is a first-generation histamine H1 receptor antagonist (Ki = 0.98 nM for the human receptor). It is selective for histamine H1 over H3 and H4 receptors (Kis = >100 and 77.6 µM, respectively, for the human receptors). Promethazine also binds muscarinic acetylcholine receptors (mAChRs, Ki = 22 nM). It...
| Keywords: | Diprazin, Fellozine, Lergigan, Phenergan, Romergan, N,N,alpha-trimethyl-10H-phenothiazine-10-ethanamine, monohydrochloride |
| Application: | H1-receptor antagonist |
| CAS | 58-33-3 |
| MW: | 320.9 D |
From 43.00€
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U-46619
Item number: Cay16450-1
U-46619 is a stable analog of the endoperoxide prostaglandin H2, and a TP receptor agonist. It exhibits properties similar to thromboxane A2, causing platelet shape change and aggregation, and contraction of vascular smooth muscle. Mean EC50 values for shape change in human, rat, and rabbit platelets are 4.8, 6.0,...
| Keywords: | 9,11-dideoxy-9alpha,11alpha-methanoepoxy PGF2alpha, 9,11-dideoxy-9alpha,11alpha-methanoepoxy Prostaglandin F2alpha,... |
| Application: | TP receptor agonist |
| CAS | 56985-40-1 |
| MW: | 350.5 D |
From 130.00€
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(±)-Taxifolin
Item number: Cay18647-500
(±)-Taxifolin is a flavonoid that has been found in M. butyracea and has diverse biological activities. It scavenges 2,2-diphenyl-1-picrylhydrazyl (DPPH, Cay-14805) radicals in cell-free assays. (±)-Taxifolin is cytotoxic to HCT116 cells (IC50 = 63.42 µM). It inhibits HMG-CoA reductase activity and cholesterol...
| Keywords: | (±)-Dihydroquercetin, (2R,3R)-rel-2-(3,4-dihydroxyphenyl)-2,3-dihydro-3,5,7-trihydroxy-4H-1-benzopyran-4-one |
| Application: | Dihyroflavonol, Lipid synthesis regulator, MMP12 inhibitor |
| CAS | 24198-97-8 |
| MW: | 304.3 D |
From 77.00€
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Picaridin
Item number: Cay16458-100
Picaridin is an insect repellent. It inhibits A. aegypti odorant receptor 2 (AaOR2) or AaOR8 in the presence of their odorant activators, indole and octenol, respectively, expressed in Xenopus oocytes (IC50s = 1,452 and 1,911 µM, respectively). Picaridin reduces the number of entries into a food chamber by female D....
| Keywords: | Bayrepel, Icaridin, KBR 3023, Saltidin(TM), 2-(2-hydroxyethyl)-1-piperidinecarboxylic acid, 1-methylpropyl ester |
| Application: | Insect repellent |
| CAS | 119515-38-7 |
| MW: | 229.3 D |
43.00€
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