4 products were found matching "Cay10007852-5"!

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Pargyline (hydrochloride)
Pargyline (hydrochloride)

Item number: Cay10007852-500

Pargyline is an irreversible inhibitor of monoamine oxidase (MAO, Kis = 15 and 1.8 µM for MAO-A and MAO-B, respectively). At 10 mg/kg i.v., pargyline induces a moderate decrease of systolic blood pressure in unanaesthetized hypertensive rats but not normotensive WKR or Sprague-Dawley rats. The correlation between...
Keywords: NSC 43798, N-methyl-N-2-propyn-1-yl-benzenemethanamine, monohydrochloride
Application: MAO inhibitor
CAS 306-07-0
MW: 195.7 D
From 14.00€ *
Review
Leukotriene E4-d5
Leukotriene E4-d5

Item number: Cay10007858-25

Leukotriene E4-d5 (LTE4-d5) contains five deuterium atoms at the 19, 19', 20, 20 and 20 positions. It is intended for use as an internal standard for the quantification of LTE4 by GC- or LC-mass spectrometry. LTE4 is produced by the action of dipeptidase on LTD4, leaving only the cysteinyl group still attached to...
Keywords: LTE4-d5, 5S-hydroxy-6R-(S-cysteinyl)-7E,9E,11Z,14Z-eicosatetraenoic-19,19,20,20,20-d5 acid
Application: Standard
CAS 1240398-14-4
MW: 444.6 D
From 390.00€ *
Review
CAY10499
CAY10499

Item number: Cay10007875-25

CAY10499 is a non-selective lipase inhibitor (IC50s = 144, 90, and 14 nM for human recombinant MAGL, HSL, and FAAH, respectively). It also inhibits ATGL, DAGLa, ABHD6, and CES1 by 95, 60, 90, and 95%, respectively, when used at a concentration of 5 mM. CAY10499 inhibits the growth of MCF-7, MDA-MB-231, COV318, and...
Keywords: [4-(5-methoxy-2-oxo-1,3,4-oxadiazol-3(2H)-yl)-2-methylphenyl]-carbamic acid, phenylmethyl ester
Application: HSL inhibitor
CAS 359714-55-9
MW: 355.3 D
From 22.00€ *
Review
(±)-Lisofylline
(±)-Lisofylline

Item number: Cay10010785-25

(±)-Lisofylline (LSF) is a potent anti-inflammatory agent in which only the (-) optical isomer is biologically active. LSF inhibits the generation of phosphatidic acid (IC50 = 0.6 µM) from cytokine-activated lysophosphatidic acyl transferase (LPAAT), which has been shown to protect mice from endotoxic shock. LSF...
Keywords: BL 194, CT-1501R, LSF, 3,7-dihydro-1-(5-hydroxyhexyl)-3,7-dimethyl-1H-purine-2,6-dione
Application: Phosphatidic acid generation inhibitor
CAS 6493-06-7
MW: 280.3 D
From 98.00€ *
Review