Palmitoyl Serotonin

Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay9000630-5 5 mg -

6 - 10 business days*

66.00€
Cay9000630-10 10 mg -

6 - 10 business days*

110.00€
Cay9000630-50 50 mg -

6 - 10 business days*

415.00€
Cay9000630-100 100 mg -

6 - 10 business days*

764.00€
 
Palmitoyl serotonin is a hybrid molecule patterned after arachidonoyl serotonin (Catalog No.... more
Product information "Palmitoyl Serotonin"
Palmitoyl serotonin is a hybrid molecule patterned after arachidonoyl serotonin (Catalog No. 70665). Arachidonoyl serotonin is a dual antagonist of fatty acid amide hydrolase (FAAH) and the transient receptor potential vanilloid-type 1 (TRPV1) channel, reducing both acute and chronic peripheral pain. The effects of replacing the arachidonoyl portion with the saturated 16-carbon palmitoyl moiety have not been studied. However, replacement of arachidonate with saturated 11- or 12-carbon fatty acids produces compounds that potently inhibit capsaicin-induced TRPV1 channel activation (IC50 = 0.76 µM) without blocking FAAH-mediated hydrolysis of arachidonoyl ethanolamine (IC50 > 50 µM).Formal Name: N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-hexadecanamide. CAS Number: 212707-51-2. Molecular Formula: C26H42N2O2. Formula Weight: 414.6. Purity: >98%. Formulation: (Request formulation change), A neat solid. Solubility: DMF: 30 mg/ml, DMSO: 15 mg/ml, Ethanol: 30 mg/ml, PBS (pH 7.2): 0.25 mg/ml. lambdamax: 223, 278 nm. SMILES: CCCCCCCCCCCCCCCC(NCCC1=CNC2=CC=C(O)C=C12)=O. InChi Code: InChI=1S/C26H42N2O2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-26(30)27-19-18-22-21-28-25-17-16-23(29)20-24(22)25/h16-17,20-21,28-29H,2-15,18-19H2,1H3,(H,27,30). InChi Key: AKQOZSXOPVLUHA-UHFFFAOYSA-N.
Keywords: N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-hexadecanamide
Supplier: Cayman Chemical
Supplier-Nr: 9000630

Properties

Application: FAAH/TRPV1 antagonist, pain studies
MW: 414.6 D
Formula: C26H42N2O2
Purity: >98%
Format: Solution

Database Information

CAS : 212707-51-2| Matching products
KEGG ID : K05222 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Signal Word: Warning
GHS Hazard Pictograms:
H Phrases: H315, H319, H335
P Phrases: P261, P264, P271, P280, P312, P321, P302+P352, P304+P340, P305+P351+P338, P332+P313, P337+P313, P362+P364, P405, P403+P233, P501
Caution
Our products are for laboratory research use only: Not for administration to humans!
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