8 products were found matching "AG-CN2-0056-C100"!
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Sipholenol A
Item number: AG-CN2-0506-C100
White to off-white lyophilized powder. Soluble in DMSO or 100% ethanol (25mg/ml). Efficient inhibitor of P-glycoprotein (Pgp, MDR-1) function through direct interactions. By inhibiting MDR-1, active compounds remain in the cytoplasm longer and allowing them to be more effective within the cell, Reversing agent for...
| Keywords: | NSC378977 |
| Application: | MDR1 inhibitor |
| CAS | 78518-73-7 |
| MW: | 476,7 D |
154.00€
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Okadaic acid (high purity)
Item number: AG-CN2-0056-C025
Non-phorbol type tumor promoter. Reversible, potent and selective serine threonine protein phosphatase inhibitor. PP2A (IC50=0. 2-1nM), PP1 (IC50=3-15nM), PP2B (IC50=>1µM). Does not inhibit PP2C. Stimulates intracellular protein phosphorylation. Useful tool for studying cellular processes that are regulated by...
| Keywords: | Halochondrine A, CCRIS 3329, HSDB 7243, 9,10-Deepithio-9,10-didehydroacanthifolicin |
| Application: | Ser/Thr phosphatase inhibitor |
| CAS | 78111-17-8 |
| MW: | 805 D |
99.00€
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Okadaic acid, ammonium salt (high purity)
Item number: AG-CN2-0058-C100
Non-phorbol type tumor promoter. Reversible, potent and selective serine threonine protein phosphatase inhibitor. PP2A (IC50=0. 2-1nM), PP1 (IC50=3-15nM), PP2B (IC50= >1µM). Does not inhibit PP2C. Stimulates intracellular protein phosphorylation. Useful tool for studying cellular processes that are regulated by...
| Keywords: | Halochondrine A, CCRIS 3329, HSDB 7243, 9,10-Deepithio-9,10-didehydroacanthifolicin |
| Application: | Ser/Thr phosphatase inhibitor |
| CAS | 155716-06-6 |
| MW: | 822 D |
From 105.00€
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Pyripyropene A
Item number: AG-CN2-0106-C250
Antibiotic, highly specific inhibitor of acyl-coenzyme A:cholesterol acetyltransferase 2 (ACAT2), anti-angiogenic, antiatherogenic and antiatherosclerotic agent. Shows cholesterol-lowering and atheroprotective activities
| Keywords: | ()-Pyripyropene A, PPPA, FO 1289A |
| Application: | ACAT2 inhibitor |
| CAS | 147444-03-9 |
| MW: | 583,2 D |
From 154.00€
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Pyranonigrin A
Item number: AG-CN2-0156-M001
Isolated from Aspergillus niger FKI-2633. Antioxidant. Radical scavenging activity towards DPPH and superoxide Shows a suppressive effect on the expression of vascular cell adhesion molecule-1 (VCAM-1) in human umbilical vein endothelial cells (HUVECs) induced by tumor necrosis factor-alpha (TNF-alpha).Insecticidal...
| Application: | Antioxidant |
| CAS | 773855-65-5 |
| MW: | 223,2 D |
From 83.00€
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Atpenin A5
Item number: AG-CN2-0100-C250
Antibiotic, antifungal, potent and specific mitochondrial complex II (succinate-ubiquinone oxidoreductase) inhibitor, mitochondrial ATP-sensitive potassium (mK(ATP)) channel activator, cardioprotective, modulates mitochondrial ROS generation during cardioprotection
| Keywords: | 3-[(2S,4S,5R)-5,6-Dichloro-2,4-dimethyl-1-oxohexyl]-4-hydroxy-5,6-dimethoxy-2(1H)-pyridinone |
| Application: | Succinate-ubiquinone oxidoreductase inhibitor |
| CAS | 119509-24-9 |
| MW: | 366,2 D |
From 143.00€
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Anomalin A
Item number: AG-CN2-0006-M001
Lck (p56lck, lymphocyte specific tyrosine kinase) inhibitor, Antioxidant, DPPH radical scavenger. Isolated from marine fungus Arthrinium sp.
| Keywords: | 2,3,6,8-Tetrahydroxy-1-methylxanthone |
| Application: | Lck inhibitor |
| CAS | 548740-86-9 |
| MW: | 274,1 D |
132.00€
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Orlistat
Item number: AG-CN2-0050-M250
Hypolipemic cell permeable and irreversible pancreatic, gastric and carboxylester lipase inhibitor. Anti-obesity and antihypercholesterolemic compound. Antitumor compound by inhibition of the thioesterase domain of fatty acid synthase (FASN). Anti-proliferative. Causes cell cycle arrest at G1 phase. Apoptosis...
| Keywords: | Tetrahydrolipstatin, Xenical, Alli, Ro-18-0647 |
| Application: | Carboxylester Lipase Inhibitor |
| Host: | Synthetic |
| CAS | 96829-58-2 |
| MW: | 495,7 D |
From 33.00€
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