3 products were found matching "Cay10011250-50"!

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NH125
NH125

Item number: Cay10011250-5

NH125 is an imidazole that has potent antibacterial properties in drug-resistant bacteria. In bacteria, NH125 inhibits several histidine kinases, inhibiting YycG with an IC50 of 6.6 µM. NH125 also decreases the viability of several cancer cell lines with IC50 values ranging from 0.7-4.7 µM. In mammalian cells, NH125...
Keywords: 1-hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium-iodide
Application: eEF-2K inhibitor
CAS 278603-08-0
MW: 524.6 D
From 54.00€ *
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CAY10577
CAY10577

Item number: Cay10011256-50

Casein kinase 2 (CK2) is a serine/threonine-selective protein kinase involved in many signal transduction pathways. CK2 is known to negatively regulate apoptosis and its activity is increased in many proliferating tissues and tumors, which lends promise as an anti-cancer drug target. CAY10577 inhibits CK2 with an...
Keywords: 7,8-dichloro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid
Application: CK2 inhibitor
CAS 300675-28-9
MW: 258.1 D
From 24.00€ *
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NSC 210902
NSC 210902

Item number: Cay10011255-50

Casein Kinase 2 (CK2) is a serine/threonine-selective protein kinase involved in many signal transduction pathways. CK2 is known to negatively regulate apoptosis, and its activity is increased in many proliferating tissues and tumors, which lends promise as an anticancer drug target. NSC 210902 inhibits CK2 with an...
Keywords: 1,4-dihydro-4-oxo-benzo[h]quinoline-3-carboxylic acid
Application: CK2 inhibitor
CAS 51726-83-1
MW: 239.2 D
From 44.00€ *
Review