9 products were found matching "Cay15734"!
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3-bromo-5-phenyl Salicylic Acid
Item number: Cay13574-1
The aldo-keto reductase (AKR) enzymes constitute a family of related NADPH-dependent oxidoreductases. The 1C subfamily (AKR1C) includes four human hydroxysteroid dehydrogenases, with AKR1C1 being a 20alpha-HSD and the other three being 3alpha-HSDs. AKR1C1 metabolizes progesterone to an inactive progestin,...
| Keywords: | NSC 109116, 5-bromo-4-hydroxy-[1,1'-biphenyl]-3-carboxylic acid |
| Application: | AKR1C1 inhibitor |
| CAS | 4906-68-7 |
| MW: | 293.1 D |
From 86.00€
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Taurolidine
Item number: Cay15374-5
Taurolidine is a synthetic taurine analog with antimicrobial and anti-neoplastic actions. It displays broad bactericidal and fungicidal activity. Taurolidine and its metabolites mimic mannose by binding to the extracellular wall of bacteria, blocking adherence to epithelial and fibroblast cells. In addition to...
| Keywords: | 4,4'-methylenebis(tetrahydro-1,2H,4-thiadiazine) 1,1,1',1'-tetraoxide |
| Application: | Antimicrobial mannose mimic |
| CAS | 19388-87-5 |
| MW: | 284.4 D |
From 43.00€
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NS 11021
Item number: Cay15347-25
NS 11021 is an activator of large-conductance Ca2+-activated potassium channels (BKCa/KCa1.1). It is selective for BKCa and is thought to bind directly the alpha subunit. NS 11021 has been shown to relax intracavernous arterial rings and corpus cavernosum strips in vitro and to enhance erectile responses in intact...
| Keywords: | N'-[3,5-bis(trifluoromethyl)phenyl]-N-[4-bromo-2-(2H-tetrazol-5-yl)phenyl]-thiourea |
| Application: | KCNMA1 activator |
| CAS | 956014-19-0 |
| MW: | 511.2 D |
From 43.00€
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Streptavidin:SureLight(TM) P3
Item number: Cay13457-1
Streptavidin conjugated to SureLight(TM) P3 Antibody: Streptavidin Dye: SureLight(TM) P3 Excitation max. lambda: 614 nm Emission max. lambda: 662 nm Uses: Flow cytometry, fluorescence-activated cell sorting, protein microarrays, and point of careEmission: 662 nm. Excitation: 614 nm. Formulation: (Request formulation...
| Application: | FC, Fluorescence |
352.00€
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Nimodipine
Item number: Cay14573-1
Nimodipine is an inhibitor of L-type voltage-gated calcium (CaV) channels. It is selective for CaV1.2 over CaV1.3 channels (IC50s = 0.139 and 2.7 µM, respectively), as well as R-, N-, and P/Q-type Cav channels at 10 µM. Nimodipine (0.72-24 nM) inhibits contractions induced by potassium, but not norepinephrine, in...
| Keywords: | BAY-e 9736, 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid, 3-(2-methoxyethyl) 5-(1-methylethyl)... |
| Application: | Ca2+ channel antagonist |
| CAS | 66085-59-4 |
| MW: | 418.4 D |
From 48.00€
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UNC0638
Item number: Cay10734-5
The methylation of lysine residues on histones plays a central role in determining euchromatin structure and gene expression. The histone methyltransferase (HMTase) G9a can mono- or dimethylate lysine 9 on histone 3 (H3), contributing to early embryogenesis, genomic imprinting, and lymphocyte development. UNC0638 is...
| Keywords: | 2-cyclohexyl-6-methoxy-N-[1-(1-methylethyl)-4-piperidinyl]-7-[3-(1-pyrrolidinyl)propoxy]-4-quinazolinamine |
| Application: | G9a HMTase inhibitor |
| CAS | 1255580-76-7 |
| MW: | 509.7 D |
From 65.00€
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DC4 Crosslinker
Item number: Cay14734-5
DC4 crosslinker is a mass spectrometry-cleavable crosslinking reagent (18Å in length) that contains two intrinsic positive charges, which allow cross-linked peptides to fragment into their component peptides by collision-induced dissociation or in-source decay. Initial fragmentation events result in cleavage on...
| Keywords: | 1,4-bis[4-[(2,5-dioxo-1-pyrrolidinyl)oxy]-4-oxobutyl]-1,4-diazoniabicyclo[2.2.2]octane, dibromide |
| Application: | MS-cleavable crosslinking reagent |
| CAS | 1374647-94-5 |
| MW: | 640.3 D |
From 85.00€
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L-ANAP methyl ester (hydrochloride)
Item number: Cay15437-10
L-ANAP methyl ester is an esterified form of the fluorescent unnatural amino acid L-ANAP (Cay-15436). It has been used in the synthesis of L-ANAP. L-ANAP methyl ester has also been used to fluorescently label proteins in vitro through genetic encoding.Formal Name: 3-[(6-acetyl-2-naphthalenyl)amino]-L-alanine, methyl...
| Keywords: | methyl (S)-3-((6-acetylnaphthalen-2-yl)amino)-2-aminopropanoate, monohydrochloride |
| Application: | Fluorescent unnatural amino acid ester |
| MW: | 322.8 D |
From 109.00€
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Trimebutine
Item number: Cay31574-5
Trimebutine is an opioid receptor agonist. It binds to µ-, delta-, and kappa-opioid receptors with Ki values of 0.34, 0.5, and 0.58 µM, respectively, in canine myenteric plexus synaptosomes. Trimebutine inhibits twitch contraction and acetylcholine (ACh) release induced by low-frequency electrical stimulation in...
| Keywords: | (±)-Trimebutine, 3,4,5-trimethoxy-benzoic acid, 2-(dimethylamino)-2-phenylbutyl ester |
| Application: | Opioid receptor agonist |
| CAS | 39133-31-8 |
| MW: | 387.5 D |
From 60.00€
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