- Search results for Cay15415
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8 products were found matching "Cay15415"!
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Item number: Cay15415-1
The histone H3 lysine 27 (H3K27) methyltransferase EZH2 plays an important role in regulating gene expression, and its aberrant activity is linked to the onset and progression of cancer. GSK126 is a selective, S-adenosyl-methionine-competitive small molecule inhibitor of EZH2 methyltransferase activity (Ki = 0.57...
Keywords: | N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-methyl-1-[(1S)-1-methylpropyl]-6-[6-(1-piperazinyl)-3-pyridinyl]-... |
Application: | Selective EZH2 methyltransferase inhibitor |
CAS | 1346574-57-9 |
MW: | 526.7 D |
From 84.00€
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Item number: Cay15411-5
cFMS kinase is the cellular homolog of the v-FMS oncogene product of the Susan McDonough strain of the feline sarcoma virus. It can autophosphorlyate colony-stimulating factor (CSF-1), which promotes the survival, proliferation, and differentiation of mononuclear phagocytes. GW 2580 selectively inhibits cFMS kinase...
Keywords: | 5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]methyl]-2,4-pyrimidinediamine |
Application: | CSF1R kinase inhibitor |
CAS | 870483-87-7 |
MW: | 366.4 D |
From 50.00€
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Item number: Cay15417-5
Modafinil (Cay-15417) is an analytical reference standard that is classified as a nootropic. It is a wake-promoting agent that binds competitively and selectively to the dopamine transporter, modulating catecholaminergic signaling by inhibiting its activity (IC50 = 3 µM, Ki = 2 µM). With much weaker potency,...
Keywords: | (±)-Modafinil, CEP-1538, CRL 40476, 2-[(diphenylmethyl)sulfinyl]-acetamide |
Application: | Analytical reference standard, Nootropic, Wake-promoting dopamine transporter inhibitor |
CAS | 68693-11-8 |
MW: | 273.4 D |
From 241.00€
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Item number: Cay15419-5
Ribonucleotide reductase, the rate-limiting enzyme for de novo DNA synthesis, is an excellent target for chemotherapy. Its increased activity in cancer cells is associated with malignant transformation and proliferation. 3-AP is a ribonucleotide reductase inhibitor and iron chelator with antitumor activity. At 5 µM...
Keywords: | 3-Aminopyridine-2-Carboxyaldehyde Thiosemicarbazone, NSC 663249, Triapine(TM),... |
Application: | Ribonucleotide reductase inhibitor |
CAS | 143621-35-6 |
MW: | 195.2 D |
From 43.00€
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Item number: Cay15410-5
PGF1beta is the C-9 epimer of PGF1alpha. It was shown to enhance respiratory rate in experimental animals when administered intravenously.Formal Name: 9beta,11alpha,15S-trihydroxy-prost-13E-en-1-oic acid. CAS Number: 10164-73-5. Synonyms: 9beta-PGF1alpha, PGF1beta. Molecular Formula: C20H36O5. Formula Weight: 356.5....
Keywords: | 9beta-PGF1alpha, PGF1beta, 9beta,11alpha,15S-trihydroxy-prost-13E-en-1-oic acid |
Application: | Bioactive lipid assays |
CAS | 10164-73-5 |
MW: | 356.5 D |
From 86.00€
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Item number: Cay15413-5
(S)-MG115 is a potent and reversible proteasome inhibitor, targeting the chymotryptic site on the 20S particle (Ki = 21 nM). It reduces the degradation of ubiquitin-conjugated proteins in extracts. (S)-MG115 also blocks the degradation of long- and short-lived proteins in intact cells as well as the proteolytic...
Keywords: | N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formylbutyl]-L-leucinamide |
Application: | Potent, reversible proteasome chymotrypsin-like activity inhibitor |
CAS | 133407-86-0 |
MW: | 461.6 D |
From 69.00€
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Item number: Cay15416-25
Pinacidil is a cyanoguanidine compound that acts as a potassium channel opener, activating the ATP-modulated potassium channels of guinea pig bladder and heart with Ki values of 104 and 251 nM, respectively. It completely relaxes coronary artery rings preconstricted with serotonin (Cay-14332, IC50 = 1.26 µM)....
Keywords: | N-cyano-N'-4-pyridinyl-N''-(1,2,2-trimethylpropyl)-guanidine, monohydrate |
CAS | 85371-64-8 |
MW: | 263.4 D |
From 39.00€
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Item number: Cay15414-25
Pitavastatin is an HMG-CoA reductase inhibitor (Ki = 1.7 nM for the rat liver microsomal enzyme). It inhibits sterol biosynthesis in rat liver and ileum (ED50s = 0.13 and 0.2 mg/kg, respectively) and reduces plasma levels of triglycerides and total cholesterol in dogs. Pitavastatin (0.3 mg/kg) increases survival in...
Keywords: | Itabastatin, Itavastatin, NK 104, (3R,5S,6E)-7-[2-cyclopropyl-4-(4-fluorophenyl)-3-quinolinyl]-3,5-dihydroxy-6-heptenoic... |
Application: | HMG-CoA reductase inhibitor |
CAS | 147526-32-7 |
MW: | 440.5 D |
From 84.00€
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