6 products were found matching "Cay15741-96"!
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4-hydroxy-3-Methoxyamphetamine (hydrochloride)
Item number: Cay14196-1
4-hydroxy-3-Methoxyamphetamine (hydrochloride) (Cay-14196) is an analytical reference standard categorized as an amphetamine. 4-hydroxy-3-Methoxyamphetamine is an active metabolite of 3,4-MDMA (Cay-ISO60190, Cay-13971, Cay-34480) via the intermediates (±)-MDA (Cay-ISO60189, Cay-11554) and 3,4-dihydroxyamphetamine...
| Keywords: | HMA, NSC 172191, 4-(2-aminopropyl)-2-methoxy-phenol, monohydrochloride |
| Application: | Analytical reference standard, amphetamine |
| CAS | 13062-61-8 |
| MW: | 217.7 D |
From 109.00€
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ML-335
Item number: Cay15196-10
The µ-opioid receptor (OPRM1) is the primary site of action for morphine and other opioids associated with the treatment of pain. The occupancy of delta-opioid receptors (OPRD1) by antagonists has been shown to enhance OPRM1 binding and signaling activity. Because heteromerization of OPRM1 and OPRD1 is thought to be...
| Keywords: | CID-23723457, CYM 51010, 1-[[4-(acetylamino)phenyl]methyl]-4-(2-phenylethyl)-4-piperidinecarboxylic acid, ethyl ester |
| Application: | OPRM1-OPRD1 heterodimerization agonist |
| CAS | 1069498-96-9 |
| MW: | 408.5 D |
From 60.00€
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25(S)-27-hydroxy Cholesterol
Item number: Cay14791-1
The liver x receptors (LXRalpha and LXRbeta) are nuclear hormone receptors whose native ligands, oxysterols, induce the expression of genes involved in cholesterol and fatty acid metabolism. 27-hydroxy Cholesterol, a sterol 27-hydroxylase-mediated cholesterol hydroxylation product, activates LXRalpha and LXRbeta in...
| Keywords: | (25S)-26-hydroxy cholesterol, (25S)-cholest-5-ene-3beta,26-diol |
| Application: | LXR alpha / beta activator |
| CAS | 56845-83-1 |
| MW: | 402.7 D |
From 77.00€
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SU 9516
Item number: Cay14796-10
SU 9516 is a 3-substituted indolinone that has anti-proliferative and pro-apoptotic activity in tumor cells. It is a potent inhibitor of several cyclin-dependent kinases (CDKs) with selectivity for Cdk2 (IC50s = 22, 40, and 200 nM for Cdk2/cyclin A, Cdk1/cyclin B, and Cdk4/cyclin D1). It does not inhibit PKC, p38,...
| Keywords: | 1,3-dihydro-3Z-(1H-imidazol-5-ylmethylene)-5-methoxy-2H-indol-2-one |
| Application: | CDK inhibitor |
| CAS | 377090-84-1 |
| MW: | 241.3 D |
From 43.00€
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JAK Inhibitor I
Item number: Cay15146-1
Janus-associated kinases (JAKs) are cytoplasmic tyrosine kinases that are required for activating the signaling of certain cytokines and growth factor receptors. JAK1 mostly activates IL-6, whereas JAK1 and JAK3 trigger IL-2 and IL-4 and JAK1 and JAK2 stimulates IFN-gamma. JAK Inhibitor I is a pyridine-containing...
| Keywords: | CMP 6, Janus-Associated Kinase Inhibitor I, Pyridone 6,... |
| Application: | JAK2, JAK3, JAK1 inhibitor |
| CAS | 457081-03-7 |
| MW: | 309.3 D |
From 39.00€
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TCS-OX2-29
Item number: Cay17419-5
Orexin receptors R1 (OX1R) and OX2R mediate the action of the neuropeptides orexin A and orexin B. TCX-OX2-29 is an antagonist of OX2R (pKi = 7.5) that exhibits >250-fold selectivity for hOX2R compared with hOX1R (IC50s = 40 nM and >10,000 nM, respectively). It blocks the inhibitory action of orexin A on...
| Keywords: | (2S)-1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-1-butanone,... |
| Application: | OX2R antagonist |
| CAS | 1610882-30-8 |
| MW: | 434 D |
From 130.00€
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