3 products were found matching "Cay15739-96"!

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PKA Inhibitor (5-24) (trifluoroacetate salt)
PKA Inhibitor (5-24) (trifluoroacetate salt)

Item number: Cay15996-1

PKI PKA Inhibitor (5-24) is a synthetic peptide inhibitor of PKA (cAMP-dependent protein kinase) (Ki = 2.3 nM) derived from the active site of the skeletal muscle inhibitor protein. It mimics the protein substrate by binding to the catalytic site through the arginine-cluster basic subsite. The prominent...
Keywords: PKI (5-24), Protein Kinase A Inhibitor (5-24),...
Application: cAMP-dependent protein kinase (PKA) inhibitor
MW: 2222.4 D
From 98.00€ *
Review
MDL 72527 (hydrochloride)
MDL 72527 (hydrochloride)

Item number: Cay13996-10

MDL 72527 is a polyamine oxidase (PAO) inhibitor that inhibits spermine oxidase and N1-acetylpolyamine oxidase (IC50s = 6.1 and 0.02 µM, respectively). It does not inhibit monoamine oxidase or D-amino acid oxidase. MDL 72527 inhibits PAO-dependent H2O2 production in vitro and in vivo and is used to study the role of...
Keywords: N1,N4-di-2,3-butadien-1-yl-1,4-butanediamine, dihydrochloride
Application: PAO inhibitor
CAS 93565-01-6
MW: 265.2 D
From 50.00€ *
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Volinanserin
Volinanserin

Item number: Cay15936-1

Volinanserin is a potent and selective antagonist of the serotonin receptor 5-HT2A (Ki = 0.36-0.85 nM). It weakly binds 5-HT2C, alpha1-adrenergic, and sigma receptors (Ki = 88, 128, and 87 nM) and much less effectively associates with other serotonin, dopamine, adrenergic, muscarinic acetylcholine receptors and...
Keywords: MDL 100907, alphaR-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol
Application: Potent, selective serotonin receptor 5-HT2A antagonist
CAS 139290-65-6
MW: 373.5 D
From 74.00€ *
Review