3 products were found matching "Cay14424"!
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Darifenacin (hydrobromide)
Item number: Cay14424-10
Darifenacin is an antagonist of M3 muscarinic acetylcholine receptors (mAChRs, Ki = 0.76 nM). It is selective for M3 over M1, M2, M4, and M5 mAChRs (Kis = 7.08, 44.67, 45.71, and 9.33 nM, respectively). Darifenacin selectively inhibits contractions in isolated guinea pig ileum, bladder, and trachea (pA2s = 9.44,...
| Keywords: | UK 88525-04, 1-[2-(2,3-dihydro-5-benzofuranyl)ethyl]-alpha,alpha-diphenyl-3-pyrrolidineacetamide, monohydrobromide |
| Application: | Muscarinic receptor antagonist |
| CAS | 133099-07-7 |
| MW: | 507.5 D |
From 92.00€
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PP1 (Src Inhibitor)
Item number: Cay14244-1
PP1 is a potent, reversible, ATP-competitive, and selective inhibitor of the Src family of protein tyrosine kinases. It inhibits p56lck (IC50 = 5 nM), p59fynT (IC50 = 6 nM), Hck (IC50 = 20 nM), and Src (IC50 = 170 nM) without significantly affecting the activity of EGFR kinase (IC50 = 250 nM), JAK2 (IC50 = 50 µM),...
| Keywords: | AGL 1872, EI 275, 1-(1,1-dimethylethyl)-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Application: | Tyrosine kinase inhibitor |
| CAS | 172889-26-8 |
| MW: | 281.4 D |
From 66.00€
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AKB48 N-pentanoic acid metabolite
Item number: Cay14224-10
AKB48 (Cay-ISO00060) is a pentyl indazole with structural similarity to JWH 018 adamantyl carboxamide (Cay-9001193) and STS-135 (Cay-11564), which are synthetic cannabinoids that may be sold for recreational use. AKB48 N-pentantoic acid metabolite is a potential urinary metabolite of AKB48, characterized by...
| Keywords: | APINACA N-pentanoic acid metabolite, 3-[(tricyclo[3.3.1.13,7]dec-1-ylamino)carbonyl]-1H-indazole-1-pentanoic acid |
| Application: | Analytical reference standard, potential urinary AKB48 metabolite |
| CAS | 1630022-94-4 |
| MW: | 395.5 D |
From 158.00€
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