7 products were found matching "Cay15981"!
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SL 327
Item number: Cay15598-1
The dual specific threonine/tyrosine kinase MEK is a key component of the RAS/RAF/MEK/ERK signaling pathway that regulates a diverse array of cellular processes. SL 327 is an inhibitor of MEK1 and MEK2 (IC50s = 0.18 and 0.22 µM), the kinases upstream of ERK1/2. It inhibits ERK1, MKK/p38, MKK4, JNK, and PKC at much...
| Keywords: | alpha-[amino[(4-aminophenyl)thio]methylene]-2-(trifluoromethyl)-benzeneacetonitrile |
| Application: | MEK1 / MEK2 inhibitor |
| CAS | 305350-87-2 |
| MW: | 335.4 D |
From 77.00€
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Lofexidine (hydrochloride)
Item number: Cay15989-1
Lofexidine is an alpha2-adrenergic receptor agonist (Kd = 7.6 nM for rat cerebral cortex membranes) that has transient antihypertensive effects. It is used in managing opioid withdrawal symptoms during detoxification from heroin (Cay-9001543) and methadone.Formal Name:...
| Keywords: | 2-[1-(2,6-dichlorophenoxy)ethyl]-4,5-dihydro-1H-imidazole, monohydrochloride |
| Application: | alpha2b-adrenergic receptor agonist |
| CAS | 21498-08-8 |
| MW: | 295.6 D |
From 54.00€
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ATM4 4-acetoxy analog
Item number: Cay15498-1
The acetylation of opium with acetic anhydride, which converts morphine to heroin, produces a variety of other acetylated products from other endogenous alkaloids, including thebaine. ATM4 4-acetoxy analog (Cay-15498) is an analytical reference standard categorized as a potential impurity in the synthesis of heroin...
| Keywords: | N-[2-[5-(acetyloxy)-3,6-dimethoxy-1-phenanthrenyl]ethyl]-N-methyl-acetamide |
| Application: | Analytical reference standard, Potential heroin synthesis impurity |
| CAS | 91295-74-8 |
| MW: | 395.5 D |
From 185.00€
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Lipid-based Drug Delivery Tools
1,2-Dioleoyl-sn-glycero-3-PC
Item number: Cay15098-1
1,2-Dioleoyl-sn-glycero-3-PC (DOPC) is a phospholipid containing the unsaturated long-chain (18:1) oleic acid inserted at the sn-1 and sn-2 positions. It is commonly used alone, or with other components, in the generation of micelles, liposomes, and other types of artificial membranes.Formal Name:...
| Keywords: | sn-3-Dioleoyllecithin, 1,2-Dioleoyl-sn-glycero-3-Phosphocholine, 1,2-DOPC, PDD 111,... |
| Application: | Phospholipid |
| CAS | 4235-95-4 |
| MW: | 786.1 D |
From 76.00€
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Stauprimide
Item number: Cay15398-1
Stauprimide is a small molecule that increases the efficiency of mouse and human embryonic stem cell differentiation in conjunction with lineage specification cues (EC50 = 0.3 µM). It specifically inhibits the nuclear localization of NME2, which results in the suppression of c-Myc, a key regulator of...
| Keywords: | N-Benzoyl-7-oxo Staurosporine,... |
| Application: | NME2 nuclear localization inhibitor |
| CAS | 154589-96-5 |
| MW: | 584.6 D |
From 68.00€
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MMP Inhibitor II
Item number: Cay15958-1
Matrix metalloproteinases (MMPs) belong to a family of proteases that play a crucial role in tissue remodeling and repair by degrading extracellular matrix proteins to enable cell migration. MMP Inhibitor II is a reversible, broad-range inhibitor of MMPs. It has been reported to inhibit MMP-1 (IC50 = 24 nM), MMP-3...
| Keywords: | Matrix Metalloproteinase Inhibitor II, NHDDPC, PG 117025, PGE 4410186,... |
| Application: | MMP-1, -3, -7, -9 inhibitor |
| CAS | 203915-59-7 |
| MW: | 513.6 D |
From 85.00€
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Edrophonium (chloride)
Item number: Cay15928-1
Edrophonium (chloride) is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by binding specifically to its catalytic site. It has been shown to inhibit AChE activity in human red blood cells, purified calf forebrain, and purified octopus brain with...
| Keywords: | Enlon(R), Tensilon(R), N-ethyl-3-hydroxy-N,N-dimethyl-benzenaminium, monochloride |
| Application: | Acetylcholinesterase (AChE) inhibitor |
| CAS | 116-38-1 |
| MW: | 201.7 D |
From 46.00€
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