6 products were found matching "Cay11178-100"!
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MAM2201 N-(4-hydroxypentyl) metabolite
Item number: Cay11778-100
MAM2201 (Cay-9001219) is a synthetic cannabinoid (CB) that is closely related, structurally, to AM2201 (Cay-10707), a compound which displays high affinities for both CB receptors. MAM2201 N-(4-hydroxypentyl) metabolite is a potential phase 1 metabolite of MAM2201, based on the known metabolism of similar compounds....
| Keywords: | [1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl](4-methyl-1-naphthalenyl)-methanone |
| Application: | Analytical reference standard, potential phase I MAM2201 metabolite |
| CAS | 1537889-05-6 |
| MW: | 389.5 D |
From 109.00€
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trans-2-Decenoic Acid
Item number: Cay17888-10
trans-2-Decenoic acid is an unsaturated fatty acid found in royal jelly produced from the hypopharyngeal and mandibular gland secretions of honeybees. It is isolated in conjunction with 10-HDA (Cay-10976) and both demonstrate weak estrogenic activity, inhibiting binding of 17beta-estradiol (Cay-ISO60155) to estrogen...
| Keywords: | trans-2-Decylenic Acid, 2E-decenoic acid |
| Application: | Estrogen receptor beta 17beta-estradiol binding inhibitor |
| CAS | 334-49-6 |
| MW: | 170.3 D |
From 98.00€
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L002
Item number: Cay17778-10
L002 is an inhibitor of p300 histone acetyltransferase (KAT3B, IC50 = 1.98 µM in vitro). It has weaker inhibitory effects against PCAF and GCN5 (IC50s = 35 and 34 µM, respectively) and is specific for p300 over a panel of additional acetyltransferases, deacetylases, and methyltransferases. L002 blocks acetylation of...
| Keywords: | NSC 764414, p300/CBP Inhibitor VI, 2,6-dimethyl-2,5-cyclohexadiene-1,4-dione 4-[O-[(4-methoxyphenyl)sulfonyl]oxime] |
| Application: | p300 histone acetyltransferase inhibitor |
| CAS | 321695-57-2 |
| MW: | 321.3 D |
From 109.00€
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BRD9539
Item number: Cay11788-10
BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 µM. It inhibits polycomb repressive complex 2 (PRC2) to a similar extent with 54 and 43% activity remaining for G9a and PRC2, respectively, when used at a concentration of 10 µM. It is selective...
| Keywords: | 2-(benzoylamino)-1-(3-phenylpropyl)-1H-benzimidazole-5-carboxylic acid |
| Application: | G9a / PRC2 inhibitor |
| CAS | 1374601-41-8 |
| MW: | 399.4 D |
From 43.00€
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GDC-0152
Item number: Cay17810-10
Inhibitor of apoptosis proteins (IAPs), which block various signaling pathways leading to apoptotic cell death, are commonly over-expressed in cancer cells. GDC-0152 is a potent inhibitor of specific IAPs that binds baculoviral IAP repeat (BIR) domains (Kis = 28, 14, 17, and 43 nM for XIAP BIR3, NL-IAP BIR, BIRC2...
| Keywords: | N-methyl-L-alanyl-(2S)-2-cyclohexylglycyl-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-L-prolinamide |
| Application: | Caspase activator |
| CAS | 873652-48-3 |
| MW: | 498.6 D |
From 60.00€
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Arachidonoyl Ethanolamide-d4
Item number: Cay10011178-100
Arachidonoyl ethanolamide-d4 (AEA-d4) contains four deuterium atoms at the hydroxyethyl 1,1',2, and 2' positions. It is intended for use as an internal standard for the quantification of AEA by GC- or LC-mass spectrometry. AEA is the ethanolamine amide of arachidonic acid, first isolated from porcine brain. It is an...
| Keywords: | AEA-d4, Anandamide-d4, N-(2-hydroxyethyl-1,1,2,2-d4)-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Application: | Standard |
| CAS | 946524-40-9 |
| MW: | 351.6 D |
From 48.00€
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