35 products were found matching "AG-CP3-0005"!
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DAMGO . acetate
Item number: AG-CP3-0005V-M001
Synthetic. Chemical. CAS: 100929-53-1. Formula: C26H35N5O6 . C2H4O2. MW: 513.6 . 60.1. Synthetic. Potent, selective agonist of µ-opioid receptor. Antinociceptive. Stimulates calcium-activated adenylyl cyclases related cAMP production. Expresses chemokines and chemokine receptors through TGF-beta1. Increases food...
| Keywords: | [D-Ala2, N-Me-Phe4, Gly5-ol]-Enkephalin, H-Tyr-D-Ala-Gly-N-Me-Phe-Gly-ol . acetate, DAGO, DAMGE, Dagol, RX 783006 |
| Application: | Potent, selective -opioid receptor agonist |
| CAS | 100929-53-1 |
| MW: | 573,7 D |
From 44.00€
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MG-132
Item number: AG-CP3-0011-M005
Soluble in DMSO or ethanol. Potent, cell permeable and selective, reversible proteasome inhibitor. Blocks degradation of short-lived proteins and induces a heat shock response. NF-kappaB activation inhibitor through IkappaB degradation. Cell permeable, reversible peptide aldehyde inhibitor. Calpain and cathepsin...
| Keywords: | Z-Leu-Leu-Leu-CHO, Z-LLL-CHO, Carbobenzoxy-L-leucyl-L-leucyl-L-leucinal, MG132 |
| Application: | Proteasome inhibitor |
| CAS | 133407-82-6 |
| MW: | 476 D |
From 22.00€
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Tirzepatide
Item number: AG-CP3-0043-M005
Tirzepatide is a novel dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist. Tirzepatide potently activates the GLP-1R signaling pathway to stimulate glucose-dependent insulin secretion through activity at the GIP receptor (GIPR) or the GLP-1R. Tirzepatide is a...
| Keywords: | LY3298176, Mounjaro |
| Application: | Glucose-dependent insulinotropic polypeptide (GIP)/glucagon-like peptide-1 (GLP-1) receptor agonist |
| CAS | 2023788-19-2 |
| MW: | 4813,5 D |
From 121.00€
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Retatrutide . sodium salt
Item number: AG-CP3-0044-M005
Retatrutide is a novel triple agonist peptide of the glucagon receptor (GCGR), glucose-dependent insulinotropic polypeptide receptor (GIPR) and glucagon-like peptide-1 receptor (GLP-1R). Retatrutide inhibits human GCGR, GIPR and GLP-1R with EC50 values of 5.79, 0.0643 and 0.775 nM, respectively and mouse GCGR, GIPR,...
| Keywords: | LY3437943, GGG Tri-agonist |
| Application: | GCGR/GIPR/GLP-1R triple agonist peptide |
| MW: | 4754.4 D |
From 132.00€
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Suc-Leu-Leu-Val-Tyr-AMC
Item number: AG-CP3-0016-M005
Solid lyophilized powder. Soluble in DMSO. Fluorogenic substrate for measuring the chymotrypsin-like peptidase activity of the 20S proteasome, calpains and other chymotrypsin-like proteases, Extinction: 380nm. Emission: 460 nm, This substrate is useful for inhibitor screening and kinetic analysis.
| Keywords: | Suc-LLVY-AMC, Proteasome Substrate, Calpain Substrate |
| Application: | Fluorogenic proteasome substrate |
| CAS | 94367-21-2 |
| MW: | 763,9 D |
From 39.00€
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Semaglutide
Item number: AG-CP3-0040-M005
Synthetic. Soluble in aqueous solution (5% AcOH) (1mg/ml). Glucagon-like peptide-1 (GLP-1) receptor agonist. Antidiabetic agent against type 2 diabetes (T2D). Stimulates insulin and suppresses glucagon secretion in a glucose-dependent manner. Longer-acting alternative to liraglutide. Chemically similar to...
| Keywords: | Semaglutide (free acid), NN 9535, NNC 0113-0217, Ozempic,... |
| Application: | Antidiabetic, Glucagon-like peptide 1 (GLP-1) receptor agonist |
| MW: | 4113.6 D |
From 66.00€
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Z-Leu-Leu-Glu-AMC
Item number: AG-CP3-0022-M005
Solid lyophilized powder. Soluble in DMSO. Fluorogenic substrate for the peptidylglutamyl-peptide hydrolysing (PGPH) (caspase-like) activity of the 20S proteasome, Excitation: 380nm. Emission: 460nm.
| Keywords: | Z-LLE-AMC, Proteasome Substrate II |
| Application: | Fluorogenic proteasome substrate |
| CAS | 348086-66-8 |
| MW: | 664,8 D |
From 44.00€
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![Z-Leu-Leu-Leu-B(OH)2 [MG-262]](https://www.biomol.com/media/image/c1/3d/5e/AG-CP3-0024-M001_200x200.png "Z-Leu-Leu-Leu-B(OH)2 [MG-262]")
Z-Leu-Leu-Leu-B(OH)2 [MG-262]
Item number: AG-CP3-0024-M005
Solid lyophilized powder. Soluble in DMSO. Highly potent and selective cell permeable inhibitor of the proteasome. Inhibits the chymotrypsin-like and caspase-like peptidase activity of the proteasome, Calpain and cathepsin inhibitor, Autophagy activator, Similar structure as MG-132 (AG-CP3-0011) but much higher...
| Keywords: | Z-LLL-B(OH)2, Proteasome Inhibitor III |
| Application: | Proteasome inhibitor |
| CAS | 179324-22-2 |
| MW: | 491,4 D |
From 77.00€
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Z-VAD-FMK (Cell permeable)
Item number: AG-CP3-0002-M005
Cell permeable, non-selective broad-spectrum caspase inhibitor. Binds irreversibly to the catalytic site of caspase proteases - The peptide is O-methylated in the P1 position on aspartic acid, providing enhanced stability and increased cell permeability - Inhibits ICE-family protease/caspase processing, leading to...
| Keywords: | Z-VAD(OMe)-FMK, pan-Caspase Inhibitor, Z-Val-Ala-DL-Asp(OMe)-fluoromethylketone,... |
| Application: | Caspase Inhibitor |
| Expressed in: | Synthetic |
| MW: | 467,5 D |
From 165.00€
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Bradykinin
Item number: AG-CP3-0025-M005
Lyophilized powder. Soluble in water (1mg/ml) or 5% acetic acid. Pro-inflammatory peptide, acting through G-protein-coupled receptors, Endogenous bradykinin receptor agonist that displays selectivity for B2 over B1 receptors, Endogenously formed following pathophysiological stimuli such as inflammation, tissue...
| Keywords: | H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH . TFA |
| Application: | Endogenous bradykinin receptor agonist |
| CAS | 121283-65-6 |
| MW: | 1174,2 D |
From 28.00€
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![Z-Leu-Leu-Nva-CHO [MG-115]](https://www.biomol.com/media/image/66/51/eb/AG-CP3-0015-M001_200x200.png "Z-Leu-Leu-Nva-CHO [MG-115]")
Z-Leu-Leu-Nva-CHO [MG-115]
Item number: AG-CP3-0015-M005
Solid lyophilized powder. Soluble in DMSO. Potent, reversible and cell permeable proteasome inhibitor. Specifically inhibits the chymotrypsin-like activity of the proteasome, Calpain and cathepsin inhibitor, Apoptosis inducer in Rat-1 and PC12 cells via a p53-dependent pathway, Autophagy activator.
| Keywords: | Z-LLNva-CHO, Proteasome Inhibitor |
| Application: | Proteasome inhibitor |
| CAS | 133407-86-0 |
| MW: | 461,6 D |
From 22.00€
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Ac-Arg-Leu-Arg-AMC
Item number: AG-CP3-0013-M005
Solid lyophilized powder. Soluble in DMSO, methanol or water (aqueous solutions). Fluorogenic tri-peptide substrate for measuring the trypsin-like peptidase activity of the 20S proteasome, It is cleaved exclusively at the amide R-AMC bond to release fluorescent product, Shows low Km and high specific activity....
| Keywords: | Ac-RLR-AMC, Proteasome Substrate |
| Application: | Proteasome substrate |
| CAS | 929903-87-7 |
| MW: | 642,8 D |
From 66.00€
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