13 products were found matching "Cay560101"!

1 from 2 pages
No results were found for the filter!
COX Inhibitor Screening Assay Potassium Hydroxide
COX Inhibitor Screening Assay Potassium Hydroxide

Item number: Cay460105-1

Synonyms: Potassium Hydroxide.
Keywords: Potassium Hydroxide
Application: COX inhibitor screening
16.00€ *
Review
Prostaglandin F2alpha
Prostaglandin F2alpha

Item number: Cay16010-5

Prostaglandin F2alpha (PGF2alpha) is a widely distributed PG occurring in many species. It causes contraction of vascular, bronchial, intestinal, and myometrial smooth muscle, and also exhibits potent luteolytic activity. PGF2alpha exerts its receptor mediated physiological activity at 50-100 nM. Maximal ovine...
Keywords: Dinoprost, PGF2alpha, 9alpha,11alpha,15S-trihydroxy-prosta-5Z,13E-dien-1-oic acid
Application: Bioactive lipid assays
CAS 551-11-1
MW: 354.5 D
From 50.00€ *
Review
Thiorphan
Thiorphan

Item number: Cay15600-10

Thiorphan is an inhibitor of neprilysin (NEP, IC50 = 0.007 µM). It selectivity inhibits NEP over NEP2 (IC50 = 22 µM), as well as angiotensin-converting enzyme (ACE) and endothelin-converting enzyme 1 (ECE1, Kis = >0.1 and >10 µM, respectively, in cell-free assays). Thiorphan (10 µM) increases bradykinin-induced...
Keywords: DL-Thiorphan, N-[2-(mercaptomethyl)-1-oxo-3-phenylpropyl]-glycine
Application: Potent neprilysin inhibitor
CAS 76721-89-6
MW: 253.3 D
From 84.00€ *
Review
R-(-)-alpha-Methylhistamine (hydrochloride)
R-(-)-alpha-Methylhistamine (hydrochloride)

Item number: Cay25601-10

R-(-)-alpha-Methylhistamine is a histamine H3 receptor agonist with diverse biological activities. It inhibits the release of histamine induced by antidromic electrical stimulation of the sciatic nerve in rats when administered at doses ranging from 0.25 to 2 mg/kg, an effect that can be reversed by the selective...
Keywords: (alphaR)-methyl-1H-imidazole-5-ethanamine, dihydrochloride
Application: Histamine H3 receptor agonist
CAS 75614-89-0
MW: 198.1 D
From 43.00€ *
Review
Indium (III) thiosemicarbazone 5b
Indium (III) thiosemicarbazone 5b

Item number: Cay35601-10

Indium (III) thiosemicarbazone 5b is an anticancer agent. It is cytotoxic to A549, MCF-7 breast, MCF-7/DDP cisplatin-resistant breast, and Hl 7702 liver cancer cells (IC50s = 2.41, 1.97, 2.11, and 8.95 µM, respectively). Indium (III) thiosemicarbazone 5b decreases PI3K, Akt, mTOR, P-gp, and GSH levels in MCF-7/DDP...
Keywords: (OC-6-43)-dichloro[N,N-dimethyl-2-[(2-pyridinyl-kappaN)methylene]hydrazinecarbothioamide-kappaN2,kappaS]methoxy-indium
Application: Anticancer agent
CAS 2345755-20-4
MW: 425 D
From 43.00€ *
Review
JWH 022
JWH 022

Item number: Cay9001056-1

JWH 022 is a cannabimimetic indole that is structurally related to JWH 018, a mildly selective agonist of the peripheral cannabinoid (CB2) receptor. The biological activity of JWH 022 has not been reported.Formal Name: 1-naphthalenyl[1-(4-penten-1-yl)-1H-indol-3-yl]-methanone. CAS Number: 209414-16-4. Molecular...
Keywords: AM2201 N-(4-pentenyl) analog, 1-naphthalenyl[1-(4-penten-1-yl)-1H-indol-3-yl]-methanone
Application: Analytical reference standard, Cannabimimetic indole (structurally related to JWH 018)
CAS 209414-16-4
MW: 339.4 D
From 241.00€ *
Review
COX (ovine/human) Inhibitor Screening Assay Kit
COX (ovine/human) Inhibitor Screening Assay Kit

Item number: Cay560131-96

The COX (ovine/human) Inhibitor Screening Assay directly measures PGF2alpha by SnCl2 reduction of COX-derived PGH2 produced in the COX reaction. The prostanoid product is quantified via enzyme immunosorbent assay (ELISA) using an antiserum specific to PGF2alpha. This assay includes both ovine COX-1 and human...
Application: COX inhibitor screening
584.00€ *
Review
Anti-Prostaglandin E Synthase (cytosolic)
Anti-Prostaglandin E Synthase (cytosolic)

Item number: Cay160150-1

Prostaglandin E synthase (PGES) catalyzes the isomerization of PGH2 (Cay-17020) to PGE2 (Cay-14010). Cytosolic and microsomal PGES enzymes have been cloned and characterized. Cytosolic PGES (cPGES) is a glutathione-dependent enzyme with a predicted size of 18.6 kDa (23 kDa on SDS-PAGE). The enzyme is expressed in a...
Keywords: Anti-P23, Anti-cPGES, Anti-cPGES, Anti-PTGES3, Anti-Hsp90 co-chaperone, Anti-Hsp90 co-chaperone, Anti-Prostaglandin E...
Application: WB
Host: Rabbit
422.00€ *
Review
Prostaglandin E Synthase (cytosolic) Blocking Peptide
Prostaglandin E Synthase (cytosolic) Blocking Peptide

Item number: Cay360150-1

Each vial contains 200 µg of lyophilized peptide derived from human cPGE synthase amino acids 58-67 (CIDPNDSKHK). This peptide was used as an antigen for production of Cayman's cPGE synthase polyclonal antibody (Catalog No. 160150) and should be used in conjunction with this antibody to block protein-antibody...
Keywords: cPGE Synthase, cPGES, Hsp90 Co-chaperone, p23, Teolomerate-binding protein p23
Application: IHC, WB
177.00€ *
Review
13,14-dihydro Prostaglandin F1alpha
13,14-dihydro Prostaglandin F1alpha

Item number: Cay15610-10

13,14-dihydro Prostaglandin F1alpha (13,14-dihydro PGF1alpha) is a potential metabolite of PGF1alpha. Its biological activity has not been reported. The corresponding compound in the E1 series (13,14-dihydro PGE1) retains biological activity similar to PGE1.Formal Name: 9alpha,11alpha,15S-trihydroxy-prostan-1-oic...
Keywords: 13,14-dihydro PGF1alpha, PGFalpha, 9alpha,11alpha,15S-trihydroxy-prostan-1-oic acid
Application: Bioactive lipid assays
CAS 20592-20-5
MW: 358.5 D
From 86.00€ *
Review
Anti-Acetyl Lysine   (Clone 7F8)
Anti-Acetyl Lysine (Clone 7F8)

Item number: Cay10010567-1

Lysine acetylation is an evolutionarily conserved posttranslational modification that is found in prokaryotes and eukaryotes at histone and non-histone protein sites. Transfer of an acetyl group from acetyl-coenzyme A (acetyl-CoA) to the amino side chain of lysine is catalyzed by lysine acetyltransferases (KATs),...
Keywords: ACE
Application: ELISA, ICC, WB
Host: Mouse
488.00€ *
Review
16-phenoxy tetranor Prostaglandin F2alpha methyl amide
16-phenoxy tetranor Prostaglandin F2alpha methyl amide

Item number: Cay10010562-1

Prostaglandin F2alpha (PGF2alpha) drives luteolysis and smooth muscle contraction by activating the FP receptor. Stable, lipophilic analogs of PGF2alpha are used to modulate luteolysis and treat glaucoma. 16-phenoxy tetranor PGF2alpha is a metabolically stable form of PGF2alpha containing a 16-phenoxy group at the...
Keywords: 16-phenoxy tetranor PGF2alpha methyl amide,...
Application: Bioactive Lipid Assays
MW: 403.5 D
From 74.00€ *
Review
1 from 2 pages