- Search results for Cay11985
Cookie preferences
This website uses cookies, which are necessary for the technical operation of the website and are always set. Other cookies, which increase the comfort when using this website, are used for direct advertising or to facilitate interaction with other websites and social networks, are only set with your consent.
Configuration
Technically required
These cookies are necessary for the basic functions of the shop.
"Allow all cookies" cookie
"Decline all cookies" cookie
CSRF token
Cookie preferences
Currency change
Customer-specific caching
FACT-Finder tracking
Individual prices
Selected shop
Session
Comfort functions
These cookies are used to make the shopping experience even more appealing, for example for the recognition of the visitor.
Note
Show the facebook fanpage in the right blod sidebar
Statistics & Tracking
Affiliate program
Conversion and usertracking via Google Tag Manager
Track device being used
11 products were found matching "Cay11985"!
Close filters
Filter by:
No results were found for the filter!
Item number: Cay11985-10
CGP 36216 is a selective antagonist of GABAB receptors (IC50 = 43 µM). Its action is reversed by the GABAB receptor agonist baclofen. It is active at presynaptic, but not postsynaptic, receptors.Formal Name: p-(3-aminopropyl)-p-ethyl-phosphinic acid, monohydrochloride. CAS Number: 1781834-71-6. Molecular Formula:...
Keywords: | p-(3-aminopropyl)-p-ethyl-phosphinic acid, monohydrochloride |
Application: | GABAB receptor antagonist |
CAS | 1781834-71-6 |
MW: | 187.6 D |
From 48.00€
*
Item number: Cay11198-5
3-Ethylethcathinone (hydrochloride) is a substituted cathinone with potential for abuse. Its biological and toxicological properties have not been evaluated. This product is intended for forensic applications.Formal Name: 2-(ethylamino)-1-(3-ethylphenyl)-1-propanone, monohydrochloride. CAS Number: 2446466-61-9....
Keywords: | 3-EEC, 2-(ethylamino)-1-(3-ethylphenyl)-1-propanone, monohydrochloride |
Application: | Analytical reference standard, Substituted cathinone with potential for abuse |
CAS | 2446466-61-9 |
MW: | 241.8 D |
From 266.00€
*
Item number: Cay19988-5
(S)-(-)-BAY-K-8644 is an activator of voltage-sensitive L-type calcium channels. It demonstrates vasoconstrictive and positive inotropic effects in vivo as well as behavioral effects, including deficits to motor function. When combined with BIX01294 (Cay-13124), (S)-(-)-BAY-K-8644 can enable reprogramming of mouse...
Keywords: | (4S)-1,4-dihydro-2,6-dimethyl-5-nitro-4-[2-(trifluoromethyl)phenyl]-3-pyridinecarboxylic acid, methyl ester |
Application: | Voltage-sensitive L-type calcium channel activator |
CAS | 98625-26-4 |
MW: | 356.3 D |
From 43.00€
*
Item number: Cay19998-5
m-Iodobenzylguanidine (MIBG) is an analogue of norepinephrine with anticancer activity. It inhibits cell growth in a panel of human and mouse leukemia, fibrosarcoma, melanoma, and neuroblastoma cell lines when used at a concentration of 20 µg/ml and reduces clonogenic survival of L1210 leukemia cells in a...
Keywords: | meta-Iodobenzylguanidine, MIBG, N-[(3-iodophenyl)methyl]-guanidine, hemisulfate |
CAS | 87862-25-7 |
MW: | 324.1 D |
From 43.00€
*
Item number: Cay11998-5
Histamine has been implicated in a variety of biological functions including thermo- and immunoregulation, food intake, hyperexcitability, pain transmission, arousal, reward, memory, and emotional responses. The histamine H3 receptor is a Gi-coupled presynaptic auto- and hetero-receptor whose activation leads to a...
Keywords: | 1-[3-[4-(1-piperidinylmethyl)phenoxy]propyl]-piperidine |
Application: | Histamine H3R antagonist |
CAS | 398473-34-2 |
MW: | 316.5 D |
From 119.00€
*
Item number: Cay11981-5
(S)-Pramipexole is a dopamine D2S, D2L, D3, and D4 receptor agonist (EC50s = 426.58, 338.84, 2.24, and 128.82 nM, respectively, in a [35S]GTPgammaS binding assay). It is also a partial agonist of alpha2A-adrenergic receptors (alpha2A-ARs, EC50 = 3,548.13 nM). (S)-Pramipexole is selective for dopamine D2-4 receptors...
Keywords: | (-)-Pramipexole, (6S)-4,5,6,7-tetrahydro-N6-propyl-2,6-benzothiazolediamine, dihydrochloride |
Application: | Galphai agonist |
CAS | 104632-25-9 |
MW: | 284.2 D |
From 43.00€
*
Item number: Cay11986-5
The metabotropic glutamate receptor 2 (mGluR2) is a Gi/o-coupled receptor which is expressed on presynaptic nerve terminals and modulates the release of neurotransmitters like glutamate and GABA. Biphenylindanone A (BINA) is a positive allosteric modulator of mGluR2, stimulating the human and rat receptors with EC50...
Keywords: | BINA, MRLSD 230, 3'-[[(2-cyclopentyl-2,3-dihydro-6,7-dimethyl-1-oxo-1H-inden-5-yl)oxy]methyl]-[1,1'-biphenyl]-4-carboxylic... |
Application: | mGluR2 modulator |
CAS | 866823-73-6 |
MW: | 454.6 D |
From 142.00€
*
Item number: Cay11989-5
Metabotropic glutamate receptors (mGluRs), mediate excitatory synaptic transmission in the central nervous system. Potent and selective antagonists of the type I mGluRs (mGluR1 and mGluR5) are of interest as novel therapeutics for the treatment of various CNS disorders, such as pain, epilepsy, and stroke. NPS 2390...
Keywords: | N-tricyclo[3.3.1.13,7]dec-1-yl-2-quinoxalinecarboxamide |
Application: | mGluR1/mGluR5 antagonist |
CAS | 226878-01-9 |
MW: | 307.4 D |
From 119.00€
*
Item number: Cay11982-5
SB 277011A is an antagonist of the dopamine D3 receptor (pKi = 8.0) that is at least 100-fold selective for D3 over other monoamine receptors (pKis = 6.0, 5.0, and 2, 5-HT1D and 5-HT1B respectively). It has high oral bioavailability and enters the central nervous system of the rat. SB 277011A has been shown to have...
Keywords: | N-[trans-4-[2-(6-cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide, dihydrochloride |
Application: | DRD3 antagonist |
CAS | 1226917-67-4 |
MW: | 511.5 D |
From 60.00€
*
Item number: Cay11983-5
Sonepiprazole is a selective antagonist of the dopamine 4 (D4) receptor (Kis = 10 nM). It is highly selective over D1, D2, and D3 receptors, serotonin 1A and 2 receptors, as well as alpha1- and alpha2-adrenergic receptors (Kis > 2,000 nM). Its safety profile in rat studies is improved in comparison to classical...
Keywords: | PNU 101387, U-101387, 4-[4-[2-[(1S)-3,4-dihydro-1H-2-benzopyran-1-yl]ethyl]-1-piperazinyl]-benzenesulfonamide |
Application: | Dopamine D4 DRD4 antagonist |
CAS | 170858-33-0 |
MW: | 401.5 D |
From 60.00€
*
Item number: Cay11984-5
Sumanirole is a dopamine D2 receptor agonist that is selective for D2 over D1, D3, and D4 receptors (Kis = 9.0, >7,140, 1,940, and >2,190 nM, respectively). It inhibits forskolin-stimulated cAMP accumulation in CHO cells expressing human recombinant D2A receptors (EC50 = 17 nM). Sumanirole decreases plasma prolactin...
Keywords: | PNU 95666, (5R)-5,6-dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one, 2Z-butenedioate |
Application: | Dopamine receptor D2 agonist |
CAS | 179386-44-8 |
MW: | 319.3 D |
From 43.00€
*