CAY10573

CAY10573
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay10008846-500 500 µg -

6 - 10 business days*

60.00€
Cay10008846-1 1 mg -

6 - 10 business days*

113.00€
Cay10008846-5 5 mg -

6 - 10 business days*

457.00€
Cay10008846-10 10 mg -

6 - 10 business days*

797.00€
 
The peroxisome proliferator-activated receptors (PPARs) are lipid-activated transcription factors... more
Product information "CAY10573"
The peroxisome proliferator-activated receptors (PPARs) are lipid-activated transcription factors often used as drug targets for the treatment of metabolic disorders. CAY10573 is a PPAR agonist that displays potent binding at PPARalpha, gamma, and delta with IC50 values of 113, 50, and 223 nM, respectively. It potently transactivates PPARalpha, gamma, and delta with EC50 values of 8, 70, and 500 nM, respectively. CAY10573 demonstrates stronger binding and functional activity for PPARgamma than the antidiabetic compound rosiglitazone (IC50 = 92 nM, EC50 = 220 nM).Formal Name: 5-[3-[(6-benzoyl-1-propyl-2-naphthalenyl)oxy]propoxy]-1H-indole-1-acetic acid. CAS Number: 853652-40-1. Molecular Formula: C33H31NO5. Formula Weight: 521.6. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 0.3 mg/ml, DMSO: 0.5 mg/ml. lambdamax: 227, 274 nm. SMILES: CCCc1c(OCCCOc2ccc3ccn(CC(=O)O)c3c2)ccc2cc(ccc12)C(=O)c1ccccc1. InChi Code: InChI=1S/C33H31NO5/c1-2-7-29-28-14-11-26(33(37)24-8-4-3-5-9-24)20-25(28)12-15-31(29)39-19-6-18-38-27-13-10-23-16-17-34(22-32(35)36)30(23)21-27/h3-5,8-17,20-21H,2,6-7,18-19,22H2,1H3,(H,35,36). InChi Key: PMPUMRAPFFYFRW-UHFFFAOYSA-N.
Keywords: 5-[3-[(6-benzoyl-1-propyl-2-naphthalenyl)oxy]propoxy]-1H-indole-1-acetic acid
Supplier: Cayman Chemical
Supplier-Nr: 10008846

Properties

Application: PPAR agonist
MW: 521.6 D
Formula: C33H31NO5
Purity: >98%
Format: Crystalline Solid

Database Information

CAS : 853652-40-1| Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
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