6 products were found matching "Cay15747-384"!
No results were found for the filter!
Norketamine (hydrochloride)
Item number: Cay15787-1
Norketamine (hydrochloride) (Cay-15787) is an analytical reference material categorized as an arylcyclohexylamine metabolite. Norketamine is a metabolite of ketamine (Cay-19389, Cay-11630). This product is intended for research and forensic applications.Formal Name: 2-amino-2-(2-chlorophenyl)-cyclohexanone,...
| Keywords: | N-desmethyl Ketamine, 2-amino-2-(2-chlorophenyl)-cyclohexanone, monohydrochloride |
| Application: | Analytical reference material, Arylcyclohexylamine metabolite |
| CAS | 79499-59-5 |
| MW: | 260.2 D |
From 43.00€
*
NS 11021
Item number: Cay15347-1
NS 11021 is an activator of large-conductance Ca2+-activated potassium channels (BKCa/KCa1.1). It is selective for BKCa and is thought to bind directly the alpha subunit. NS 11021 has been shown to relax intracavernous arterial rings and corpus cavernosum strips in vitro and to enhance erectile responses in intact...
| Keywords: | N'-[3,5-bis(trifluoromethyl)phenyl]-N-[4-bromo-2-(2H-tetrazol-5-yl)phenyl]-thiourea |
| Application: | KCNMA1 activator |
| CAS | 956014-19-0 |
| MW: | 511.2 D |
From 43.00€
*
Galiellalactone
Item number: Cay15387-1
Galiellalactone is a fungal metabolite isolated from the ascomycetes G. rufa strain A75-86 and A111-95 that inhibits IL-6-mediated JAK/STAT signal transduction in HepG2 cells with an IC50 value of 0.25-0.5 µM. The selectivity of this compound is achieved by its ability to block the binding of activated STAT3 dimers...
| Keywords: | (7bS)-5,5aR,6,7,7aR,7b-hexahydro-7b-hydroxy-4S-methyl-indeno[1,7-bc]furan-2(4H)-one |
| Application: | JAK/STAT signal transduction inhibitor |
| CAS | 133613-71-5 |
| MW: | 194.2 D |
From 294.00€
*
STAT5 Inhibitor
Item number: Cay15784-5
Signal Transducers and Activators of Transcriptions (STATs) are a family of cytoplasmic latent transcription factors that are activated to regulate gene expression in response to a large number of extracellular signaling polypeptides including cytokines, interferons, and growth factors. STAT5, which consists of two...
| Keywords: | Signal Transducers and Activators of Transcription 5, 2-[(4-oxo-4H-1-benzopyran-3-yl)methylene]hydrazide... |
| Application: | Cell permeable STAT5 inhibitor |
| CAS | 285986-31-4 |
| MW: | 293.3 D |
From 92.00€
*
Bicyclomycin Benzoate
Item number: Cay15384-5
Bicyclomycin benzoate is an antibiotic produced by S. sapporonensis that inhibits Gram-negative bacteria, including E. coli, Klebsiella, Shigella, Salmonella, Citrobacter, E. cloacae, and the pathogenic group of Neisseria. It is inactive against Proteus, P. aeruginosa, and Gram-positive bacteria.Formal Name:...
| Keywords: | FR2054, 3'-benzoate bicyclomycin |
| Application: | Antibiotic |
| CAS | 37134-40-0 |
| MW: | 406.4 D |
From 189.00€
*
AZD 8186
Item number: Cay17384-1
AZD 8186 is a selective PI3Kbeta/delta inhibitor that exhibits IC50 values of 3, 17, and 752 nM for PI3Kbeta, delta, and alpha, respectively, in cells sensitive to isoform-specific PI3K inhibition. It shows no significant binding against a panel of 442 other kinases when tested at a concentration of 10 µM and...
| Keywords: | 8-[(1R)-1-[(3,5-difluorophenyl)amino]ethyl]-N,N-dimethyl-2-(4-morpholinyl)-4-oxo-4H-1-benzopyran-6-carboxamide |
| Application: | PI3Kbeta/delta inhibitor |
| CAS | 1627494-13-6 |
| MW: | 457.5 D |
From 43.00€
*